SCHEMBL20972

SCHEMBL20972

CNC(=O)C1(OCCOC)CCC(c2nc3c(-c4cnn(-c5ccccc5)c4)cnn3c(N)c2SC)CC1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 10/20 0.35
CCNA2 P20248 10/20 0.35
CDK2 P24941 10/20 0.35
CCNA1 P78396 10/20 0.35
GRM4 Q14833 5/20 0.34
TYK2 P29597 1/20 0.34
TTK P33981 1/20 0.33
CCNC P24863 1/20 0.33
CDK8 P49336 1/20 0.33
RET P07949 1/20 0.33
KIF5B P33176 1/20 0.33
KDR P35968 1/20 0.33
ETV6 P41212 1/20 0.33
KCNH2 Q12809 1/20 0.33
CCDC6 Q16204 1/20 0.33
GRM2 Q14416 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15006972 0.93 CHEK1 (0.37) CHEK1CCNA2CDK2CCNA1GRM4
SCHEMBL20640 0.93 CHEK1 (0.37) CHEK1CCNA2CDK2CCNA1GRM4
SCHEMBL21922 0.93 CHEK1 (0.37) CHEK1CCNA2CDK2CCNA1GRM4
SCHEMBL15007359 0.92 CFTR (0.34) CHEK1CCNA2CDK2CCNA1GRM4
SCHEMBL15007311 0.91 CHEK1 (0.35) CHEK1CCNA2CDK2CCNA1GRM4
SCHEMBL15006919 0.89 CHEK1 (0.34) CHEK1CCNA2CDK2CCNA1GRM4
SCHEMBL15031480 0.89 CHEK1 (0.34) CHEK1CCNA2CDK2CCNA1GRM4
SCHEMBL15006918 0.89 CHEK1 (0.34) CHEK1CCNA2CDK2CCNA1GRM4
SCHEMBL15007221 0.88 CHEK1 (0.34) CHEK1CCNA2CDK2CCNA1GRM4
SCHEMBL22015 0.88 CHEK1 (0.34) CHEK1CCNA2CDK2CCNA1GRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012027236-A1 NOVEL PYRAZOLO[1,5-a]PYRIMIDINE DERIVATIVES AS mTOR INHIBITORS SCHERING CORPORATION (US) 2012-03-01 WO disclosed