SCHEMBL20998600

SCHEMBL20998600

C=CC(=O)N1C[C@@H]2C1CN2c1ncc(C(N)=O)c(Oc2ccc(Oc3ccccc3)cc2)n1

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BTK Q06187 20/20 0.57
CYP2C8 P10632 1/20 0.57
KCNH2 Q12809 1/20 0.57
EGFR P00533 1/20 0.43
TEC P42680 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16676735 1.00 BTK (0.57) BTKCYP2C8KCNH2EGFRTEC
SCHEMBL18044913 0.86 BTK (0.74) BTKCYP2C8KCNH2EGFRTEC
SCHEMBL16670060 0.85 BTK (0.65) BTKCYP2C8KCNH2EGFRTEC
SCHEMBL21100914 0.85 BTK (0.75) BTKCYP2C8KCNH2EGFRTEC
SCHEMBL20998672 0.85 BTK (0.75) BTKCYP2C8KCNH2EGFRTEC
SCHEMBL20998573 0.85 BTK (0.75) BTKCYP2C8KCNH2EGFRTEC
SCHEMBL16676816 0.85 BTK (0.75) BTKCYP2C8KCNH2EGFRTEC
SCHEMBL16676786 0.85 BTK (0.75) BTKCYP2C8KCNH2EGFRTEC
SCHEMBL18070180 0.84 BTK (0.42) BTKCYP2C8KCNH2
SCHEMBL16676741 0.84 BTK (0.42) BTKCYP2C8KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3060550-B1 HETEROARYL COMPOUNDS AS BTK INHIBITORS AND USES THEREOF MERCK PATENT GMBH (DE) 2019-05-15 EP disclosed