SCHEMBL21031868

SCHEMBL21031868

Cc1ccc2c(c1)c(-c1csc3ccc(C(F)(F)F)cc13)c(C)n2CC(=O)O

nearest known ligand 0.66

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 19/20 0.66
PTGS1 P23219 2/20 0.48
CYP2C9 P11712 1/20 0.48
SLC6A4 P31645 1/20 0.48
CYP2C19 P33261 1/20 0.48
PTGS2 P35354 1/20 0.48
AKR1B1 P15121 2/20 0.46
AKR1A1 P14550 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21032723 0.92 PTGDR2 (0.66) PTGDR2PTGS1CYP2C9SLC6A4CYP2C19
SCHEMBL24179996 0.92 PTGDR2 (0.60) PTGDR2CYP2C9AKR1B1
SCHEMBL21031946 0.88 PTGDR2 (0.53) PTGDR2PTGS1CYP2C9SLC6A4CYP2C19
SCHEMBL21031945 0.85 PTGDR2 (0.63) PTGDR2PTGS1CYP2C9SLC6A4CYP2C19
SCHEMBL24180036 0.85 PTGDR2 (0.63) PTGDR2PTGS1CYP2C9SLC6A4CYP2C19
SCHEMBL21032143 0.85 PTGDR2 (0.61) PTGDR2PTGS1AKR1B1
SCHEMBL21032469 0.84 PTGDR2 (0.60) PTGDR2CYP2C9AKR1B1
SCHEMBL21031929 0.83 PTGDR2 (0.64) PTGDR2PTGS1CYP2C9SLC6A4CYP2C19
SCHEMBL24179951 0.83 PTGDR2 (0.56) PTGDR2CYP2C9AKR1B1
SCHEMBL21032474 0.83 PTGDR2 (0.61) PTGDR2PTGS1AKR1B1AKR1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3489233-A1 INDOLE DERIVATIVE USED AS CRTH2 INHIBITOR Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2019-05-29 EP disclosed