SCHEMBL21032465

SCHEMBL21032465

Cc1c(Cc2ccc3c(n2)C(F)(F)CC[S+]3[O-])c2cc(F)ccc2n1CC(=O)O

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 20/20 0.58
PTGDR Q13258 2/20 0.58
PTGIR P43119 1/20 0.58
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C8 P10632 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2A6 P11509 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2B6 P20813 1/20 0.50
CYP2C19 P33261 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21186600 0.83 PTGDR2 (0.58) PTGDR2
SCHEMBL24179998 0.81 PTGDR2 (0.62) PTGDR2PTGDRPTGIRCYP1A2CYP3A4
SCHEMBL21031852 0.81 PTGDR2 (0.64) PTGDR2PTGDRPTGIRCYP1A2CYP3A4
SCHEMBL21032176 0.79 PTGDR2 (0.69) PTGDR2PTGDRPTGIR
SCHEMBL16210801 0.75 PTGDR2 (0.54) PTGDR2
SCHEMBL1786702 0.75 PTGDR2 (0.85) PTGDR2PTGDRPTGIRCYP1A2CYP3A4
SCHEMBL24180051 0.75 PTGDR2 (0.52) PTGDR2
Timapiprant SCHEMBL29648518 0.74 PTGDR2 (1.00) PTGDR2PTGDRPTGIRCYP1A2CYP3A4
Timapiprant SCHEMBL29379400 0.74 PTGDR2 (1.00) PTGDR2PTGDRPTGIRCYP1A2CYP3A4
Timapiprant SCHEMBL1782956 0.74 PTGDR2 (1.00) PTGDR2PTGDRPTGIRCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3489233-A1 INDOLE DERIVATIVE USED AS CRTH2 INHIBITOR Chia Tai Tianqing Pharmaceutical Group Co., Ltd. (CN) 2019-05-29 EP disclosed