SCHEMBL21055964

SCHEMBL21055964

O=C(C1CCS(=O)(=O)CC1)N1CCN(c2ccc(OCCCN3CCCCC3)cc2)CC1

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 14/20 0.61
KCNH2 Q12809 2/20 0.58
MAOB P27338 1/20 0.54
MAPT P10636 2/20 0.52
ALDH1A1 P00352 1/20 0.52
GAA P10253 1/20 0.52
HRH2 P25021 2/20 0.51
HRH1 P35367 2/20 0.51
POLB P06746 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3580433 0.91 HRH3 (0.66) HRH3KCNH2MAOBMAPTALDH1A1
SCHEMBL6472573 0.80 HRH3 (0.72) HRH3KCNH2MAPTALDH1A1GAA
SCHEMBL3586173 0.79 HRH3 (0.71) HRH3KCNH2MAOBMAPTALDH1A1
Hydrochloric Acid SCHEMBL3581152 0.78 HRH3 (0.69) HRH3KCNH2MAPTALDH1A1GAA
SCHEMBL3581520 0.78 HRH3 (0.62) HRH3KCNH2MAOBMAPTALDH1A1
SCHEMBL21659403 0.78 HRH3 (0.68) HRH3KCNH2MAOBMAPTALDH1A1
SCHEMBL3585244 0.77 HRH3 (0.71) HRH3KCNH2MAPTALDH1A1GAA
Hydrochloric Acid SCHEMBL5935422 0.77 HRH3 (0.67) HRH3MAOBHRH2HRH1
Hydrochloric Acid SCHEMBL5935373 0.77 HRH3 (0.67) HRH3MAOBHRH2HRH1
SCHEMBL14006880 0.76 HRH3 (0.98) HRH3KCNH2HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3057963-B1 PIPERAZINE DERIVATIVES AND THE USE THEREOF AS MEDICAMENT BOEHRINGER INGELHEIM INT (DE) 2019-06-19 EP disclosed