SCHEMBL21065130

SCHEMBL21065130

FC(F)(F)Oc1ccccc1-c1cc([C@@H]2CCCN2)on1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 1/20 0.45
HCRTR2 O43614 1/20 0.45
S1PR1 P21453 2/20 0.42
SCN9A Q15858 6/20 0.40
ACP1 P24666 1/20 0.39
CNR2 P34972 1/20 0.38
TACR1 P25103 1/20 0.38
TRPA1 O75762 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28214769 0.83 HCRTR1 (0.48) HCRTR1HCRTR2S1PR1SCN9ACNR2
Hydrochloric Acid SCHEMBL30605726 0.82 HCRTR1 (0.48) HCRTR1HCRTR2S1PR1SCN9ACNR2
Hydrochloric Acid SCHEMBL21065175 0.81 HCRTR1 (0.45) HCRTR1HCRTR2S1PR1SCN9AACP1
SCHEMBL16463722 0.78 HCRTR1 (0.46) HCRTR1HCRTR2S1PR1SCN9AACP1
SCHEMBL16463721 0.78 HCRTR1 (0.46) HCRTR1HCRTR2S1PR1SCN9AACP1
SCHEMBL21065081 0.78 NR1H4 (0.55) HCRTR1HCRTR2S1PR1
SCHEMBL21065075 0.77 S1PR1 (0.49) HCRTR1HCRTR2S1PR1
Hydrochloric Acid SCHEMBL17064071 0.77 HCRTR1 (0.45) HCRTR1HCRTR2S1PR1SCN9AACP1
Hydrochloric Acid SCHEMBL17064070 0.77 HCRTR1 (0.45) HCRTR1HCRTR2S1PR1SCN9AACP1
SCHEMBL16464687 0.75 NPC1 (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2906553-B1 OREXIN RECEPTOR ANTAGONISTS WHICH ARE [ORTHO BI (HETERO )ARYL]-[2-(META BI (HETERO)ARYL)-PYRROLIDIN-1-YL]-METHANONE DERIVATIVES IDORSIA PHARMACEUTICALS LTD (CH) 2019-06-26 EP disclosed