SCHEMBL21065142

SCHEMBL21065142

COc1ccccc1-c1nnc(C2CCCN2C(=O)OC(C)(C)C)[nH]1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.44
ALDH1A1 P00352 3/20 0.44
LMNA P02545 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
HCRTR1 O43613 8/20 0.44
HCRTR2 O43614 8/20 0.44
EPHX2 P34913 1/20 0.42
SCD5 Q86SK9 1/20 0.42
GCK P35557 1/20 0.42
MAPT P10636 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
CCNT1 O60563 1/20 0.40
CDK9 P50750 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21065140 1.00 TSHR (0.44) TSHRALDH1A1LMNAMEN1KMT2A
SCHEMBL21065228 0.89 HCRTR1 (0.46) TSHRALDH1A1LMNAMEN1KMT2A
SCHEMBL17063849 0.89 HCRTR1 (0.51) HCRTR1HCRTR2
SCHEMBL21065230 0.89 HCRTR1 (0.46) TSHRALDH1A1LMNAMEN1KMT2A
SCHEMBL17063850 0.89 HCRTR1 (0.51) HCRTR1HCRTR2
SCHEMBL21065054 0.84 HCRTR1 (0.46) TSHRALDH1A1LMNAHCRTR1HCRTR2
SCHEMBL21065150 0.84 TSHR (0.49) TSHRALDH1A1LMNAMEN1KMT2A
SCHEMBL21065056 0.84 HCRTR1 (0.46) TSHRALDH1A1LMNAHCRTR1HCRTR2
SCHEMBL21065149 0.84 TSHR (0.49) TSHRALDH1A1LMNAMEN1KMT2A
SCHEMBL4956602 0.84 TSHR (0.47) TSHRALDH1A1LMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2906553-B1 OREXIN RECEPTOR ANTAGONISTS WHICH ARE [ORTHO BI (HETERO )ARYL]-[2-(META BI (HETERO)ARYL)-PYRROLIDIN-1-YL]-METHANONE DERIVATIVES IDORSIA PHARMACEUTICALS LTD (CH) 2019-06-26 EP disclosed