SCHEMBL21075880

SCHEMBL21075880

CN/C(=C\C=N)Nc1nccc(-c2cc3c(s2)C(C)(C)N(CCN2CCCOCC2)C3=O)n1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK3 P27361 1/20 0.62
MAPK1 P28482 1/20 0.62
EIF2AK2 P19525 1/20 0.34
CCNB2 O95067 1/20 0.34
CDK1 P06493 1/20 0.34
CCNB1 P14635 1/20 0.34
CCNB3 Q8WWL7 1/20 0.34
CASR P41180 1/20 0.33
MAPK13 O15264 1/20 0.33
MAPK12 P53778 1/20 0.33
MAPK11 Q15759 1/20 0.33
MAPK14 Q16539 1/20 0.33
ABL1 P00519 1/20 0.33
BCR P11274 1/20 0.33
MKNK1 Q9BUB5 1/20 0.33
GSK3B P49841 2/20 0.32
EGFR P00533 2/20 0.32
WNT1 P04628 1/20 0.32
DYRK1A Q13627 1/20 0.32
MKNK2 Q9HBH9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21075927 0.97 MAPK1 (0.66) MAPK3MAPK1EIF2AK2CCNB2CDK1
SCHEMBL21075882 0.90 MAPK1 (0.56) MAPK3MAPK1EIF2AK2CCNB2CDK1
SCHEMBL21075925 0.90 MAPK3 (0.56) MAPK3MAPK1IKBKBCHUKIKBKG
SCHEMBL21075891 0.90 MAPK3 (0.56) MAPK3MAPK1EIF2AK2CCNB2CDK1
SCHEMBL21075872 0.90 MAPK3 (0.56) MAPK3MAPK1EIF2AK2CCNB2CDK1
SCHEMBL21075977 0.89 MAPK3 (0.55) MAPK3MAPK1MAPK13MAPK12MAPK11
SCHEMBL21075890 0.87 MAPK3 (0.52) MAPK3MAPK1
SCHEMBL21075999 0.87 MAPK3 (0.53) MAPK3MAPK1
SCHEMBL21075929 0.87 MAPK3 (0.53) MAPK3MAPK1GSK3BWNT1DYRK1A
SCHEMBL21075870 0.86 MAPK3 (0.52) MAPK3MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3237423-B1 THIENO[2,3-C]PYRROL-4-ONE DERIVATIVES AS ERK INHIBITORS LILLY CO ELI (US) 2019-06-05 EP disclosed