SCHEMBL2108260

SCHEMBL2108260

CCCCCCn1sc(Cl)c(Cl)c1=O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KAT2B Q92831 3/20 0.61
MGLL Q99685 5/20 0.50
FAAH O00519 3/20 0.50
ALDH1A1 P00352 1/20 0.45
TP53 P04637 1/20 0.45
HSP90AA1 P07900 1/20 0.45
CYP3A4 P08684 1/20 0.45
G6PD P11413 1/20 0.45
HPGD P15428 1/20 0.45
ALOX15 P16050 1/20 0.45
TSHR P16473 1/20 0.45
HIF1A Q16665 1/20 0.45
HSD17B10 Q99714 1/20 0.45
RGS4 P49798 5/20 0.41
RGS8 P57771 4/20 0.41
PTGS1 P23219 3/20 0.39
PTGS2 P35354 3/20 0.39
GSK3B P49841 1/20 0.35
TNF P01375 1/20 0.35
GBA1 P04062 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8445189 1.00 KAT2B (0.61) KAT2BMGLLFAAHALDH1A1TP53
SCHEMBL13837721 1.00 KAT2B (0.61) KAT2BMGLLFAAHALDH1A1TP53
SCHEMBL8445220 1.00 KAT2B (0.61) KAT2BMGLLFAAHALDH1A1TP53
SCHEMBL204793 1.00 KAT2B (0.61) KAT2BMGLLFAAHALDH1A1TP53
SCHEMBL8444108 1.00 KAT2B (0.61) KAT2BMGLLFAAHALDH1A1TP53
SCHEMBL8444183 1.00 KAT2B (0.61) KAT2BMGLLFAAHALDH1A1TP53
SCHEMBL8444180 1.00 KAT2B (0.61) KAT2BMGLLFAAHALDH1A1TP53
Hydrochloric Acid SCHEMBL9130658 0.98 KAT2B (0.59) KAT2BMGLLFAAHALDH1A1TP53
SCHEMBL8440674 0.98 KAT2B (0.63) KAT2BMGLLFAAHALDH1A1TP53
SCHEMBL8444109 0.93 KAT2B (0.66) KAT2BMGLLFAAHALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 30 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5912286-A Silicone-containing fluoropolymers for controlled release of organic leachants THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE NAVY (US) 1999-06-15 US claimed
EP-0762955-A4 ANTIFOULING AND FOUL-RELEASE COATINGS US HEALTH (US) 1998-01-07 EP claimed
EP-0762955-A1 ANTIFOULING AND FOUL-RELEASE COATINGS THE GOVERNMENT OF THE UNITED STATES OF AMERICA, as represented by THE SECRETARY OF THE NAVY (US) 1997-03-19 EP claimed
WO-1995032862-A1 ANTIFOULING AND FOUL-RELEASE COATINGS THE GOVERNMENT OF THE UNITED STATES OF AMERICA, REPRESENTED BY THE SECRETARY OF THE NAVY (US) 1995-12-07 WO claimed
EP-0147970-B1 MICROBIOCIDAL OR ANTIMICROBIAL BIOMEDICAL DEVICES ROHM AND HAAS COMPANY (US) 1989-03-01 EP claimed
US-4542169-A Biomedical devices containing isothiazolones to control bacteria growth ROHM AND HAAS COMPANY (US) 1985-09-17 US claimed
EP-0147970-A1 Microbiocidal or antimicrobial biomedical devices ROHM AND HAAS COMPANY (US) 1985-07-10 EP claimed
US-4127687-A PAINTING WITH ISOTHIAZOLONES ROHM AND HAAS COMPANY (US) 1978-11-28 US claimed
US-8157877-B2 Chemical mechanical polishing aqueous dispersion, chemical mechanical polishing method, and kit for preparing chemical mechanical polishing aqueous dispersion JSR CORPORATION (JP) 2012-04-17 US disclosed
US-20090325323-A1 AQUEOUS DISPERSION FOR CHEMICAL MECHANICAL POLISHING, PRODUCTION METHOD THEREOF, AND CHEMICAL MECHANICAL POLISHING METHOD JSR CORPORATION (JP) 2009-12-31 US disclosed
US-20090165395-A1 CHEMICAL MECHANICAL POLISHING AQUEOUS DISPERSION, CHEMICAL MECHANICAL POLISHING METHOD, AND KIT FOR PREPARING CHEMICAL MECHANICAL POLISHING AQUEOUS DISPERSION JSR CORPORATION (JP) 2009-07-02 US disclosed
EP-1962334-A1 AQUEOUS DISPERSION FOR CHEMICAL MECHANICAL POLISHING, CHEMICAL MECHANICAL POLISHING METHOD, AND KIT FOR PREPARING AQUEOUS DISPERSION FOR CHEMICAL MECHANICAL POLISHING JSR Corporation (JP) 2008-08-27 EP disclosed
US-6786944-B2 FOR USE IN MICRO ISOLATING STEP OR A PLANARIZING STEP OF AN INTER LAYER DIELECTRIC IN PRODUCTION OF SEMICONDUCTOR DEVICES JSR CORPORATION (JP) 2004-09-07 US disclosed
EP-1357161-A2 Aqueous dispersion for chemical mechanical polishing JSR Corporation (JP) 2003-10-29 EP disclosed
EP-0410726-B1 S-SUBSTITUTED BETA-THIOACRYLAMIDES AND THEIR USE AS MICROBICIDES ROHM AND HAAS COMPANY (US) 1993-09-01 EP disclosed
US-5118681-A Bactericides ROHM AND HAAS COMPANY (US) 1992-06-02 US disclosed
EP-0410726-A1 S-substituted beta-thioacrylamides and their use as microbicides ROHM AND HAAS COMPANY (US) 1991-01-30 EP disclosed
EP-0147970-B1 MICROBIOCIDAL OR ANTIMICROBIAL BIOMEDICAL DEVICES ROHM AND HAAS COMPANY (US) 1989-03-01 EP disclosed
US-4542169-A Biomedical devices containing isothiazolones to control bacteria growth ROHM AND HAAS COMPANY (US) 1985-09-17 US disclosed
EP-0147970-A1 Microbiocidal or antimicrobial biomedical devices ROHM AND HAAS COMPANY (US) 1985-07-10 EP disclosed