SCHEMBL2108489

SCHEMBL2108489

CC(C)(C)N(C(=O)O)C1=N[C@@]2(c3cc(N)ccc3F)CC[C@@H](F)C[C@H]2CS1.CC(C)(C)N(C(=O)O)C1=N[C@@]2(c3cc(N)ccc3F)CC[C@@H](F)C[C@H]2CS1

nearest known ligand 0.36

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.36
BACE2 Q9Y5Z0 4/20 0.36
KCNH2 Q12809 2/20 0.34
CYP2D6 P10635 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2110303 1.00 BACE1 (0.36) BACE1BACE2KCNH2CYP2D6
SCHEMBL2108493 1.00 BACE1 (0.36) BACE1BACE2KCNH2CYP2D6
SCHEMBL2108109 1.00 BACE1 (0.36) BACE1BACE2KCNH2CYP2D6
SCHEMBL2108012 1.00 BACE1 (0.36) BACE1BACE2KCNH2CYP2D6
SCHEMBL2110418 0.91 BACE1 (0.36) BACE1BACE2KCNH2CYP2D6
SCHEMBL2108685 0.91 BACE1 (0.36) BACE1BACE2KCNH2CYP2D6
SCHEMBL2110416 0.91 BACE1 (0.36) BACE1BACE2KCNH2CYP2D6
SCHEMBL2109255 0.89 BACE1 (0.35) BACE1BACE2KCNH2CYP2D6
SCHEMBL2108021 0.89 BACE1 (0.35) BACE1BACE2KCNH2CYP2D6
SCHEMBL2107010 0.89 BACE1 (0.35) BACE1BACE2KCNH2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8158620-B2 Fused aminodihydrothiazine derivatives EISAI R&D MANAGEMENT CO., LTD. (JP) 2012-04-17 US disclosed