SCHEMBL21089291

SCHEMBL21089291

CN(Cc1ccccc1CBr)C(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 3/20 0.43
SLC6A4 P31645 3/20 0.43
AKT1 P31749 2/20 0.42
RIPK1 Q13546 2/20 0.41
GLS O94925 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
SOS1 Q07889 1/20 0.38
PDK2 Q15119 1/20 0.37
CTSL P07711 1/20 0.37
CTSB P07858 1/20 0.37
CTSS P25774 1/20 0.37
CACNA1G O43497 1/20 0.37
CACNA1B Q00975 1/20 0.37
CACNA1C Q13936 1/20 0.37
MEN1 O00255 1/20 0.37
CRHBP P24387 1/20 0.37
KMT2A Q03164 1/20 0.37
CRHR2 Q13324 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8017533 0.92 HTR2C (0.47) HTR2CSLC6A4AKT1RIPK1GLS
SCHEMBL18173003 0.86 AKT1 (0.43) HTR2CSLC6A4AKT1RIPK1CYP1A2
SCHEMBL15261600 0.84 HTR2C (0.43) HTR2CSLC6A4AKT1RIPK1CYP1A2
SCHEMBL7408449 0.84 HTR2C (0.43) HTR2CSLC6A4AKT1RIPK1GLS
SCHEMBL29430479 0.83 HTR2C (0.45) HTR2CSLC6A4AKT1RIPK1GLS
SCHEMBL11470297 0.83 HTR2C (0.45) HTR2CSLC6A4AKT1RIPK1GLS
SCHEMBL30264826 0.83 HSP90AA1 (0.47) HTR2CSLC6A4RIPK1GLSPDK2
SCHEMBL22687996 0.82 HTR2C (0.44) HTR2CSLC6A4AKT1RIPK1GLS
SCHEMBL1399434 0.81 HTR2C (0.43) HTR2CSLC6A4AKT1RIPK1GLS
SCHEMBL2061803 0.81 SLC6A4 (0.43) HTR2CSLC6A4AKT1RIPK1GLS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3286172-B1 LSD1 INHIBITORS AND USES THEREOF CONSTELLATION PHARMACEUTICALS INC (US) 2019-06-12 EP disclosed