SCHEMBL21097102

SCHEMBL21097102

COC(=O)c1cnc2nc(C)sc2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 9/20 0.49
RAB9A P51151 9/20 0.49
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
RXFP1 Q9HBX9 2/20 0.49
ATM Q13315 1/20 0.45
PSMD14 O00487 1/20 0.42
MAPK1 P28482 2/20 0.41
PIK3CA P42336 1/20 0.41
PIK3CB P42338 1/20 0.41
PIK3CG P48736 1/20 0.41
PI4KB Q9UBF8 1/20 0.41
HDAC1 Q13547 1/20 0.40
SMN1; SMN2 Q16637 5/20 0.40
KDM4E B2RXH2 3/20 0.40
ALDH1A1 P00352 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
PDGFRB P09619 2/20 0.39
KDR P35968 2/20 0.39
CYP2A6 P11509 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21096506 0.85 CYP2C9 (0.47) NPC1RAB9AMEN1KMT2ARXFP1
SCHEMBL20031275 0.83 NPC1 (0.53) NPC1RAB9AMEN1KMT2ARXFP1
SCHEMBL21061889 0.81 NPC1 (0.41) NPC1RAB9AMEN1KMT2ARXFP1
SCHEMBL20489431 0.81 SMN1; SMN2 (0.45) NPC1RAB9AMEN1KMT2ARXFP1
SCHEMBL21061845 0.81 NPC1 (0.41) NPC1RAB9AMEN1KMT2ARXFP1
SCHEMBL21061882 0.79 NPC1 (0.42) NPC1RAB9AATMPSMD14MAPK1
SCHEMBL21061808 0.79 NPC1 (0.40) NPC1RAB9AMEN1KMT2ARXFP1
SCHEMBL21061887 0.77 NPC1 (0.41) NPC1RAB9AATMPSMD14MAPK1
SCHEMBL23350442 0.75 MAPK1 (0.44) NPC1RAB9AMEN1KMT2AATM
SCHEMBL20375538 0.74 CYP2A6 (0.39) NPC1RAB9AMEN1KMT2AATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019116256-A1 FUSED PYRIDINES WHICH ACT AS INHIBITORS OF H-PGDS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2019-06-20 WO disclosed