SCHEMBL21099229

SCHEMBL21099229

CCCC(=O)N(C=O)OC(=O)CCCOc1ccc2c(c1)CCC/C2=N\NC(=O)CC(C)(C)S

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.41
GAA P10253 3/20 0.40
LMNA P02545 2/20 0.40
GRK2 P25098 3/20 0.39
ROCK2 O75116 2/20 0.39
MAPT P10636 7/20 0.39
HTT P42858 1/20 0.39
MEN1 O00255 1/20 0.37
BRD4 O60885 1/20 0.36
SMN1; SMN2 Q16637 3/20 0.34
POLB P06746 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
ALDH1A1 P00352 1/20 0.33
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21098772 0.96 BRD4 (0.39) KMT2AGAALMNAGRK2ROCK2
SCHEMBL21098936 0.93 KMT2A (0.40) KMT2AGAALMNAGRK2ROCK2
SCHEMBL22802047 0.83 MAPT (0.46) KMT2AGAALMNAGRK2ROCK2
SCHEMBL22802046 0.83 MAPT (0.46) KMT2AGAALMNAGRK2ROCK2
SCHEMBL21098730 0.83 MAPT (0.46) KMT2AGAALMNAGRK2ROCK2
SCHEMBL21052018 0.81 MAPT (0.44) KMT2AGAALMNAGRK2ROCK2
SCHEMBL21052015 0.81 MAPT (0.44) KMT2AGAALMNAGRK2ROCK2
SCHEMBL21098753 0.81 MAPT (0.44) KMT2AGAALMNAGRK2ROCK2
SCHEMBL21098749 0.80 SMN1; SMN2 (0.42) KMT2AGAALMNAGRK2ROCK2
SCHEMBL21052174 0.80 SMN1; SMN2 (0.42) KMT2AGAALMNAGRK2ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019109188-A1 ACYL HYDRAZONE LINKERS, METHODS AND USES THEREOF ONTARIO INSTITUTE FOR CANCER RESEARCH (OICR) (CA) 2019-06-13 WO disclosed