SCHEMBL21099403

SCHEMBL21099403

COc1cccc(F)c1-c1c(Cl)cc2c3c(cnc2c1F)OC[C@H]1CN(C(=O)OC(C)(C)C)[C@H](C)CN31

nearest known ligand 0.53

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KRAS P01116 12/20 0.53
TNF P01375 4/20 0.36
LITAF Q99732 4/20 0.36
RPS6KA1 Q15418 1/20 0.35
NTRK1 P04629 1/20 0.34
MAP4K1 Q92918 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21100011 0.91 KRAS (0.64) KRASRPS6KA1
SCHEMBL21050759 0.91 KRAS (0.57) KRASRPS6KA1NTRK1MAP4K1
SCHEMBL21099583 0.89 KRAS (0.63) KRASTNFLITAF
SCHEMBL21099226 0.85 KRAS (0.66) KRASRPS6KA1
SCHEMBL21099328 0.85 KRAS (0.55) KRASRPS6KA1
SCHEMBL21100010 0.84 KRAS (0.46) KRASTNFLITAFNTRK1
SCHEMBL21099210 0.83 KRAS (0.65) KRASTNFLITAF
SCHEMBL21099615 0.83 KRAS (0.43) KRASTNFLITAFNTRK1MAP4K1
SCHEMBL23137433 0.82 KRAS (0.40) KRASTNFLITAFNTRK1MAP4K1
SCHEMBL23137440 0.82 KRAS (0.39) KRASTNFLITAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20190177338-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2019-06-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190177338-A1 CHEMICAL COMPOUNDS MKI67, CCNI, MCL1 KRAS 272/4885TNF 2176/4885LITAF 995/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.