SCHEMBL21101258

SCHEMBL21101258

CC(=O)c1cnc2c(-c3cc(Cl)cc(Cl)c3)cccc2c1N(C)C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSA P10619 2/20 0.37
RAB9A P51151 3/20 0.36
NPC1 O15118 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
POLB P06746 1/20 0.36
GPBAR1 Q8TDU6 2/20 0.36
NUDT1 P36639 1/20 0.35
CNR2 P34972 2/20 0.35
GAA P10253 1/20 0.35
TSHR P16473 1/20 0.35
HAVCR2 Q8TDQ0 1/20 0.35
MAPT P10636 1/20 0.34
ATF1 P18846 1/20 0.34
NFKB1 P19838 1/20 0.34
KDM4E B2RXH2 1/20 0.34
HPGD P15428 1/20 0.34
GRIN2B Q13224 1/20 0.34
KCNA5 P22460 1/20 0.34
BTK Q06187 1/20 0.33
PRKAG1 P54619 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29440739 0.92 HAVCR2 (0.42) CTSAGPBAR1NUDT1CNR2HAVCR2
SCHEMBL21101077 0.92 HAVCR2 (0.42) CTSAGPBAR1NUDT1CNR2HAVCR2
Hydrochloric Acid SCHEMBL28436307 0.91 HAVCR2 (0.41) CTSAGPBAR1NUDT1CNR2HAVCR2
Hydrochloric Acid SCHEMBL30853500 0.91 HAVCR2 (0.41) CTSAGPBAR1NUDT1CNR2HAVCR2
SCHEMBL22118244 0.88 ATF1 (0.38) CTSAGPBAR1NUDT1CNR2ATF1
SCHEMBL20702326 0.86 MEN1 (0.47) SMN1; SMN2POLBMAPTKDM4E
SCHEMBL22118278 0.81 SSTR2 (0.36) GPBAR1NUDT1MAPT
SCHEMBL22118251 0.80 MEN1 (0.39) NPC1SMN1; SMN2GAAMAPTKDM4E
SCHEMBL20154226 0.79 CNR2 (0.41) SMN1; SMN2POLBCNR2MAPTKDM4E
SCHEMBL22135011 0.79 SSTR2 (0.34) GPBAR1NUDT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019115768-A1 PROCESS FOR PREPARING ANTIHELMINTIC 4-AMINO-QUINOLINE-3-CARBOXAMIDE DERIVATIVES BAYER ANIMAL HEALTH GMBH (DE) 2019-06-20 WO disclosed