SCHEMBL21101968

SCHEMBL21101968

COc1ccc(-c2nc3c(C)ccnc3[nH]2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.54
TNKS O95271 2/20 0.54
TNKS2 Q9H2K2 2/20 0.54
GSK3A P49840 9/20 0.54
GSK3B P49841 9/20 0.54
CCNB2 O95067 9/20 0.54
CDK1 P06493 9/20 0.54
CCNB1 P14635 9/20 0.54
CCNB3 Q8WWL7 9/20 0.54
CDK5 Q00535 7/20 0.54
CDK5R1 Q15078 7/20 0.54
AURKA O14965 1/20 0.49
CCNE1 P24864 1/20 0.46
CDK2 P24941 1/20 0.46
ZAP70 P43403 1/20 0.46
PTK2B Q14289 1/20 0.46
RIPK1 Q13546 1/20 0.46
KDM4E B2RXH2 1/20 0.46
NPC1 O15118 1/20 0.46
ALDH1A1 P00352 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17236527 0.82 TNKS (0.52) PARP1TNKSTNKS2GSK3AGSK3B
SCHEMBL4148211 0.82 MGAM (0.57) TNKSTNKS2GSK3AGSK3BCCNB2
SCHEMBL4157363 0.82 MGAM (0.57) TNKSTNKS2GSK3BAURKAKDM4E
SCHEMBL17224938 0.82 TNKS (0.49) PARP1TNKSTNKS2
SCHEMBL1665479 0.81 TNKS (0.51) PARP1TNKSTNKS2
SCHEMBL4941364 0.81 MAPK14 (0.52) PARP1TNKSTNKS2GSK3AGSK3B
SCHEMBL15972177 0.80 PRMT5 (0.67)
SCHEMBL4160756 0.80 PARP1 (0.50) PARP1GSK3AGSK3BCCNB2CDK1
SCHEMBL3927381 0.78 TNKS (0.55) PARP1TNKSTNKS2GSK3AGSK3B
SCHEMBL15972383 0.78 PRMT5 (0.67)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2804859-B1 NOVEL FAP INHIBITORS UNIV ANTWERPEN (BE) 2019-06-12 EP disclosed