SCHEMBL21112974

SCHEMBL21112974

CCc1ccc(/C=C/C(N)Cc2ccccc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.45
SLC6A2 P23975 2/20 0.43
TAAR1 Q96RJ0 2/20 0.43
SLC6A4 P31645 2/20 0.43
MAOA P21397 1/20 0.43
SLC6A3 Q01959 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
CYP2A6 P11509 1/20 0.43
ADORA2A P29274 1/20 0.43
ADORA1 P30542 1/20 0.43
EPHX1 P07099 1/20 0.41
CYP2D6 P10635 1/20 0.41
PPARG P37231 1/20 0.40
PPARA Q07869 1/20 0.40
ALOX5 P09917 1/20 0.38
PTGS1 P23219 1/20 0.38
PTGS2 P35354 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21065984 0.86 EPHX1 (0.50) SLC6A2TAAR1SLC6A4MAOASLC6A3
SCHEMBL13733263 0.86 EPHX1 (0.50) SLC6A2TAAR1SLC6A4MAOASLC6A3
SCHEMBL15521920 0.86 EPHX1 (0.50) SLC6A2TAAR1SLC6A4MAOASLC6A3
SCHEMBL12525245 0.86 EPHX1 (0.50) SLC6A2TAAR1SLC6A4MAOASLC6A3
SCHEMBL13733261 0.86 EPHX1 (0.50) SLC6A2TAAR1SLC6A4MAOASLC6A3
SCHEMBL12524560 0.86 EPHX1 (0.50) SLC6A2TAAR1SLC6A4MAOASLC6A3
SCHEMBL12525249 0.79 MAOB (0.48) NPC1LMNAMAPTHTTRAB9A
SCHEMBL7307677 0.76 EPHX1 (0.61) SLC6A2TAAR1SLC6A4MAOASLC6A3
SCHEMBL902538 0.76 EPHX1 (0.61) SLC6A2TAAR1SLC6A4MAOASLC6A3
SCHEMBL2736329 0.76 EPHX1 (0.61) SLC6A2TAAR1SLC6A4MAOASLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3501546-A2 CYSTEINE DRUG CONJUGATES AND USE OF SAME Seattle Genetics, Inc. (US) 2019-06-26 EP disclosed