SCHEMBL21118372

SCHEMBL21118372

Fc1ccc(I)c(-n2nccn2)c1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 18/20 0.35
HCRTR2 O43614 18/20 0.35
CYP1A2 P05177 1/20 0.35
KCNN4 O15554 1/20 0.33
KCNA5 P22460 1/20 0.33
CA3 P07451 1/20 0.31
CA6 P23280 1/20 0.31
CA5A P35218 1/20 0.31
CA9 Q16790 1/20 0.31
CA14 Q9ULX7 1/20 0.31
CA5B Q9Y2D0 1/20 0.31
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20551535 0.76 NPC1 (0.36) HCRTR1HCRTR2CYP3A4
SCHEMBL14886152 0.76 HCRTR1 (0.40) HCRTR1HCRTR2CYP1A2
SCHEMBL21894128 0.73 HCRTR1 (0.43) HCRTR1HCRTR2CYP1A2
SCHEMBL4550945 0.72 HCRTR1 (0.41) HCRTR1HCRTR2CYP1A2
SCHEMBL13647699 0.72 HCRTR1 (0.33) HCRTR1HCRTR2CYP1A2KCNN4KCNA5
SCHEMBL18195993 0.72 HCRTR2 (0.36) HCRTR1HCRTR2CYP1A2
SCHEMBL14883243 0.72 ALK (0.39) HCRTR1HCRTR2CYP1A2
SCHEMBL20781056 0.72 KDM4E (0.39) HCRTR1HCRTR2CYP1A2
SCHEMBL2523972 0.72 HCRTR2 (0.39) HCRTR1HCRTR2
SCHEMBL27900612 0.72 HCRTR2 (0.49) HCRTR1HCRTR2CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3115362-B1 PIPERIDINE DERIVATIVES AS OREXIN RECEPTOR ANTAGONIST SHANGHAI HAIYAN PHARMACEUTICAL TECH CO LTD (CN) 2019-06-12 EP disclosed