SCHEMBL21118622

SCHEMBL21118622

N=C/C=N\Nc1cc(F)ccc1C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.43
GAA P10253 5/20 0.43
RAB9A P51151 5/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
NFKB1 P19838 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43
CLCN2 P51788 1/20 0.41
GRIK1 P39086 3/20 0.40
KEAP1 Q14145 1/20 0.39
MAPT P10636 3/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 2/20 0.39
HPGD P15428 1/20 0.39
ALOX12 P18054 1/20 0.39
TRPA1 O75762 1/20 0.35
KCNK2 O95069 1/20 0.35
CES2 O00748 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23616124 0.84 CLCN2 (0.44) NPC1GAARAB9ACLCN2GRIK1
SCHEMBL23616119 0.79 AKR1C3 (0.55) NPC1GAARAB9AMEN1KMT2A
SCHEMBL19902996 0.78 KMT2A (0.52) NPC1GAARAB9ASMN1; SMN2MAPT
SCHEMBL22383441 0.77 GAA (0.45) NPC1GAARAB9ASMN1; SMN2NFKB1
SCHEMBL20976784 0.75 CHRNA4 (0.42)
SCHEMBL14555058 0.74 HCRTR2 (0.36)
SCHEMBL21118611 0.73 KDM4E (0.51) SMN1; SMN2ALDH1A1KDM4EMPO
SCHEMBL22365614 0.73 MEN1 (0.47) MAPTMEN1KMT2AALDH1A1HPGD
SCHEMBL16482031 0.72 GAA (0.43) NPC1GAARAB9ASMN1; SMN2NFKB1
SCHEMBL3810854 0.71 CLCN2 (0.52) GAACLCN2GRIK1KEAP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3115362-B1 PIPERIDINE DERIVATIVES AS OREXIN RECEPTOR ANTAGONIST SHANGHAI HAIYAN PHARMACEUTICAL TECH CO LTD (CN) 2019-06-12 EP disclosed