SCHEMBL21132528

SCHEMBL21132528

Cc1ccc(CNS(=O)(=O)c2ccc(NC(=O)NCc3cccnc3)cc2)cc1

nearest known ligand 0.80

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 16/20 0.80
ALDH1A1 P00352 1/20 0.74
MAPT P10636 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL163267 0.92 NAMPT (0.80) NAMPTMAPT
SCHEMBL29635698 0.92 NAMPT (0.80) NAMPTMAPT
SCHEMBL161983 0.91 NAMPT (0.81) NAMPTMAPT
SCHEMBL164981 0.90 NAMPT (0.83) NAMPT
SCHEMBL29635869 0.90 NAMPT (0.83) NAMPT
SCHEMBL23747377 0.90 NAMPT (0.78) NAMPT
SCHEMBL166387 0.90 NAMPT (0.78) NAMPT
SCHEMBL15310921 0.90 NAMPT (0.78) NAMPT
SCHEMBL29635822 0.90 NAMPT (0.78) NAMPT
SCHEMBL165205 0.89 NAMPT (0.84) NAMPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10329275-B2 Compounds and compositions for the inhibition of NAMPT FORMA TM, LLC (US) 2019-06-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10329275-B2 Compounds and compositions for the inhibition of NAMPT NAMPT, NNT, NQO1 NAMPT 1/4885ALDH1A1 511/4885MAPT 694/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.