SCHEMBL21135586

SCHEMBL21135586

CNC(=O)c1ccccc1Nc1nc(Nc2ccc3c(c2OC)CCC[C@H](N2CCN(C)CC2)C3)ncc1Cl

nearest known ligand 0.89

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 19/20 0.89
INSR P06213 16/20 0.89
PTK2 Q05397 12/20 0.89
KCNH2 Q12809 5/20 0.66
MET P08581 2/20 0.60
MAP4K1 Q92918 1/20 0.59
IGF1R P08069 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cep-37440 SCHEMBL29489150 0.94 ALK (1.00) ALKINSRPTK2KCNH2MET
Cep-37440 SCHEMBL15272087 0.94 ALK (1.00) ALKINSRPTK2KCNH2MET
Cep-37440 SCHEMBL16571623 0.94 ALK (1.00) ALKINSRPTK2KCNH2MET
Cep-37440 SCHEMBL31579317 0.94 ALK (1.00) ALKINSRPTK2KCNH2MET
Cep-37440 SCHEMBL29354193 0.94 ALK (1.00) ALKINSRPTK2KCNH2MET
Cep-37440 SCHEMBL15269443 0.94 ALK (1.00) ALKINSRPTK2KCNH2MET
SCHEMBL16570664 0.94 ALK (0.83) ALKINSRPTK2KCNH2MET
Cep-37440 SCHEMBL15269779 0.93 ALK (0.99) ALKINSRPTK2KCNH2MET
SCHEMBL16571176 0.93 ALK (0.91) ALKINSRPTK2KCNH2MET
SCHEMBL23810091 0.93 ALK (0.82) ALKINSRPTK2KCNH2MET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019113071-A1 COMPOSITIONS AND METHODS FOR TREATING ALK-MEDIATED CANCER ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI (US) 2019-06-13 WO disclosed