SCHEMBL21156530

SCHEMBL21156530

Cc1c(C(=O)O)cc2cc(-c3ccc(CN4CCOCC4)cc3)cn2c1C(C)N1CCOCC1

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
EED O75530 17/20 0.53
RBBP4 Q09028 17/20 0.53
SUZ12 Q15022 17/20 0.53
EZH2 Q15910 17/20 0.53
AEBP2 Q6ZN18 17/20 0.53
HRH3 Q9Y5N1 2/20 0.43
DHODH Q02127 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21156121 0.90 EED (0.52) EEDRBBP4SUZ12EZH2AEBP2
SCHEMBL21156559 0.89 EED (0.50) EEDRBBP4SUZ12EZH2AEBP2
SCHEMBL21113197 0.88 EED (0.52) EEDRBBP4SUZ12EZH2AEBP2
SCHEMBL21156102 0.87 EED (0.53) EEDRBBP4SUZ12EZH2AEBP2
SCHEMBL21156099 0.87 EED (0.64) EEDRBBP4SUZ12EZH2AEBP2
SCHEMBL21113287 0.85 EED (0.52) EEDRBBP4SUZ12EZH2AEBP2
SCHEMBL21157285 0.85 EED (0.51) EEDRBBP4SUZ12EZH2AEBP2
SCHEMBL19964844 0.84 EED (0.48) EEDRBBP4SUZ12EZH2AEBP2
SCHEMBL21156524 0.82 EED (0.49) EEDRBBP4SUZ12EZH2AEBP2
SCHEMBL21156564 0.81 EED (0.51) EEDRBBP4SUZ12EZH2AEBP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109790160-B Pyrido five-membered aromatic ring compound, preparation method and application thereof 上海海和药物研究开发股份有限公司 2022-11-15 CN disclosed
US-10968215-B2 Pyrido five-element aromatic ring compound, preparation method therefor and use thereof SHANGHAI HAIHE PHARMACEUTICAL CO., LTD. (CN) 2021-04-06 US disclosed
US-20190211010-A1 PYRIDO FIVE-ELEMENT AROMATIC RING COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF HAIHE BIOPHARMA CO. LTD. (CN) 2019-07-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10968215-B2 Pyrido five-element aromatic ring compound, preparation method therefor and use thereof EZH2, IKZF2, SUZ12 EED 41/4885RBBP4 288/4885SUZ12 3/4885
US-20190211010-A1 PYRIDO FIVE-ELEMENT AROMATIC RING COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF EZH2, IKZF2, SUZ12 EED 41/4885RBBP4 288/4885SUZ12 3/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.