SCHEMBL21170664

SCHEMBL21170664

CN(C)CCCOc1cc(F)c(-c2c(S)nc(-c3cnccn3)nc2Cl)c(F)c1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.41
LIMK1 P53667 9/20 0.36
LIMK2 P53671 8/20 0.36
MAPT P10636 1/20 0.34
CHRNB2 P17787 2/20 0.33
CHRNA4 P43681 2/20 0.33
CYP2D6 P10635 2/20 0.33
CYP2C9 P11712 2/20 0.33
CYP2C19 P33261 2/20 0.33
CYP19A1 P11511 1/20 0.33
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CXCR1 P25024 1/20 0.31
MAPK14 Q16539 1/20 0.31
ALOX5 P09917 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4018558 0.83 LIMK1 (0.37) HRH3LIMK1LIMK2MAPT
SCHEMBL15626293 0.81 LIMK1 (0.36) HRH3LIMK1LIMK2MAPK14
SCHEMBL16989331 0.81 LIMK1 (0.36) HRH3LIMK1LIMK2MAPK14
SCHEMBL4020442 0.80 LIMK1 (0.36) HRH3LIMK1LIMK2
SCHEMBL4019006 0.78 LIMK1 (0.37) HRH3LIMK1LIMK2MAPTCHRNB2
SCHEMBL21170636 0.77 NPC1 (0.43) MAPTCYP2D6CYP2C9CYP2C19CYP19A1
SCHEMBL13870028 0.74 HRH3 (0.36) HRH3LIMK1LIMK2
SCHEMBL4019009 0.73 LIMK1 (0.36) LIMK1LIMK2
SCHEMBL13901881 0.72 NPC1 (0.40) LIMK1LIMK2
SCHEMBL13870032 0.72 LIMK1 (0.34) HRH3LIMK1LIMK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2903436-B1 HETEROCYCLIC COMPOUNDS AND THEIR USE FOR THE TREATMENT OF NEURODEGENERATIVE TAUOPATHIES UNIV PENNSYLVANIA (US) 2019-07-17 EP disclosed