SCHEMBL21187109

SCHEMBL21187109

CC(=O)NC(C)C1CCC(c2ccnc3ccc(F)cc23)CC1

nearest known ligand 0.76

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 20/20 0.76
CYP2C9 P11712 3/20 0.74
CYP2C8 P10632 2/20 0.74
CHRNA1 P02708 1/20 0.74
CYP2C19 P33261 1/20 0.74
CYP3A4 P08684 1/20 0.62
TDO2 P48775 1/20 0.62
KCNH2 Q12809 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20905247 1.00 IDO1 (0.76) IDO1CYP2C9CYP2C8CHRNA1CYP2C19
SCHEMBL20916336 0.91 IDO1 (0.76) IDO1CYP2C9CYP2C8CHRNA1CYP2C19
SCHEMBL20916344 0.91 IDO1 (0.76) IDO1CYP2C9CYP2C8CHRNA1CYP2C19
SCHEMBL20916333 0.91 IDO1 (0.76) IDO1CYP2C9CYP2C8CHRNA1CYP2C19
SCHEMBL23801484 0.89 IDO1 (0.75) IDO1CYP2C9CYP2C8CHRNA1CYP2C19
SCHEMBL20956235 0.89 IDO1 (0.90) IDO1CYP2C9CYP2C8CHRNA1CYP2C19
SCHEMBL20905250 0.89 IDO1 (0.90) IDO1CYP2C9CYP2C8CHRNA1CYP2C19
SCHEMBL17746339 0.89 IDO1 (0.89) IDO1CYP2C9CYP2C8CHRNA1CYP2C19
SCHEMBL17746338 0.89 IDO1 (0.89) IDO1CYP2C9CYP2C8CHRNA1CYP2C19
SCHEMBL20905191 0.88 IDO1 (0.94) IDO1CYP2C9CYP2C8CHRNA1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141095-A1 AMIDINE AND GUANIDINE DERIVATIVE, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 四川科伦博泰生物医药股份有限公司 2019-07-25 WO disclosed