SCHEMBL21187339

SCHEMBL21187339

Cc1ncnc2cc(N3CCOCC3)cc(O[C@H]3CC[C@@H](NC(=O)OC(C)(C)C)CC3)c12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 2/20 0.38
ERBB2 P04626 2/20 0.38
BTK Q06187 3/20 0.37
CACNB4 O00305 1/20 0.36
CACNA1A O00555 1/20 0.36
CACNA1G O43497 1/20 0.36
CACNG3 O60359 1/20 0.36
CACNA1F O60840 1/20 0.36
CACNA1H O95180 1/20 0.36
CACNB3 P54284 1/20 0.36
CACNA2D1 P54289 1/20 0.36
CACNG7 P62955 1/20 0.36
CACNA1B Q00975 1/20 0.36
CACNA1D Q01668 1/20 0.36
CACNB1 Q02641 1/20 0.36
CACNG1 Q06432 1/20 0.36
CACNB2 Q08289 1/20 0.36
CACNA1S Q13698 1/20 0.36
CACNA1C Q13936 1/20 0.36
CACNA1E Q15878 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21178579 0.90 RAF1 (0.40) MAP4K4ERBB2BTKCACNB4CACNA1A
SCHEMBL21187398 0.90 RAF1 (0.40) MAP4K4ERBB2BTKCACNB4CACNA1A
SCHEMBL21187338 0.89 JAK3 (0.41) MAP4K4BTKCACNB4CACNA1ACACNA1G
SCHEMBL21178350 0.89 JAK3 (0.41) MAP4K4BTKCACNB4CACNA1ACACNA1G
SCHEMBL21187340 0.84 IRAK4 (0.38) ERBB2TBK1JAK2
SCHEMBL21279209 0.83 CACNB4 (0.39) MAP4K4BTKCACNB4CACNA1ACACNA1G
SCHEMBL16079597 0.83 CACNB4 (0.39) MAP4K4BTKCACNB4CACNA1ACACNA1G
SCHEMBL21178721 0.82 CACNB4 (0.38) MAP4K4BTKCACNB4CACNA1ACACNA1G
SCHEMBL21187263 0.82 CKS1B (0.39) ERBB2BTKCACNB4CACNA1ACACNA1G
SCHEMBL21178132 0.82 CKS1B (0.39) ERBB2BTKCACNB4CACNA1ACACNA1G

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019143678-A1 DNA-PK INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2019-07-25 WO disclosed