SCHEMBL21188141

SCHEMBL21188141

Cc1nocc1-c1ccc2c(-c3nc(NC4CCC(C)(C)NC4)ncc3C(F)(F)F)nn(PI)c2n1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCNK O75909 18/20 0.51
CDK12 Q9NYV4 18/20 0.51
CCNE1 P24864 16/20 0.51
CDK2 P24941 16/20 0.51
CCNT1 O60563 14/20 0.51
CDK9 P50750 14/20 0.51
CDK7 P50613 10/20 0.51
CCNH P51946 10/20 0.51
MNAT1 P51948 6/20 0.49
CYP2D6 P10635 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24087380 1.00 CCNK (0.51) CCNKCDK12CCNE1CDK2CCNT1
SCHEMBL21188571 0.86 CCNK (0.47) CCNKCDK12CCNE1CDK2CCNT1
SCHEMBL21188592 0.84 CCNK (0.64) CCNKCDK12CCNE1CDK2CCNT1
SCHEMBL21179179 0.84 CCNK (0.54) CCNKCDK12CCNE1CDK2CCNT1
SCHEMBL21179184 0.84 CCNK (0.54) CCNKCDK12CCNE1CDK2CCNT1
SCHEMBL24087252 0.77 CCNK (0.70) CCNKCDK12CCNE1CDK2CCNT1
SCHEMBL21188575 0.76 RXFP1 (0.30)
SCHEMBL24087469 0.76 CCNK (0.55) CCNKCDK12CCNE1CDK2CCNT1
SCHEMBL24087399 0.75
SCHEMBL21188146 0.72 CCNK (0.76) CCNKCDK12CCNE1CDK2CCNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019143719-A1 INHIBITORS OF CYCLIN-DEPENDENT KINASE 7 (CDK7) SYROS PHARMACEUTICALS, INC. (US) 2019-07-25 WO disclosed