SCHEMBL21190842

SCHEMBL21190842

Cc1cc(Br)n2nc[nH]c(=O)c12

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 4/20 0.50
PARP1 P09874 5/20 0.33
NR1H2 P55055 1/20 0.32
HPGD P15428 1/20 0.32
HTT P42858 1/20 0.31
CHEK1 O14757 2/20 0.30
PIM1 P11309 2/20 0.30
ALDH1A1 P00352 1/20 0.30
AKT1 P31749 1/20 0.30
FLT3 P36888 1/20 0.30
PIM3 Q86V86 1/20 0.30
PDPK1 O15530 1/20 0.30
RPS6KA3 P51812 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4044142 0.82 BRD4 (0.49) BRD4PARP1NR1H2HPGDHTT
SCHEMBL5816653 0.72 BRD4 (0.36) BRD4NR1H2HPGDALDH1A1
SCHEMBL16210384 0.72 PDE2A (0.38) BRD4PARP1NR1H2HPGDALDH1A1
SCHEMBL24458506 0.69 NR1H2 (0.43) BRD4PARP1NR1H2HPGDALDH1A1
SCHEMBL12365544 0.69 BRD4 (0.39) BRD4PARP1NR1H2CHEK1PIM1
SCHEMBL12365567 0.69 BRD4 (0.39) BRD4PARP1NR1H2HPGDHTT
SCHEMBL18168816 0.68 BRD4 (0.32) BRD4HPGD
SCHEMBL18742167 0.68 PDE2A (0.40) BRD4NR1H2ALDH1A1
SCHEMBL12365546 0.67 BRD4 (0.40) BRD4PARP1NR1H2ALDH1A1
SCHEMBL21190756 0.67 BRD4 (1.00) BRD4PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141131-A1 BROMODOMAIN INHIBITOR COMPOUND AND USE THEREOF 中国科学院上海药物研究所 2019-07-25 WO disclosed
US-9359548-B2 Organic electroluminescent device UDC IRELAND LIMITED (IE) 2016-06-07 US disclosed