SCHEMBL21191007

SCHEMBL21191007

Nc1ccc(OC2CCOCC2)c(Br)c1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SYK P43405 1/20 0.44
RAF1 P04049 1/20 0.39
BRAF P15056 1/20 0.39
PDE4D Q08499 6/20 0.39
PDE4A P27815 5/20 0.39
PDE4B Q07343 5/20 0.39
PDE4C Q08493 5/20 0.39
KAT2B Q92831 1/20 0.38
BAZ2B Q9UIF8 1/20 0.38
TBK1 Q9UHD2 5/20 0.35
CSNK2A1 P68400 2/20 0.35
VEGFA P15692 1/20 0.34
KDM4E B2RXH2 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
PIK3CA P42336 1/20 0.34
IKBKE Q14164 3/20 0.33
IKBKB O14920 1/20 0.33
CHUK O15111 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20021966 0.85 CSNK2A1 (0.44) PDE4DPDE4APDE4BPDE4CCSNK2A1
SCHEMBL20384187 0.83 CSNK2A1 (0.43) PDE4DPDE4APDE4BPDE4CCSNK2A1
SCHEMBL19527744 0.83 SYK (0.47) SYKRAF1BRAFPDE4DPDE4A
SCHEMBL20443368 0.81 MCHR1 (0.43) PDE4ACSNK2A1KDM4EGAAMAPT
SCHEMBL24252789 0.81 SYK (0.44) SYKPDE4DPDE4APDE4BPDE4C
SCHEMBL30986494 0.80 SYK (0.40) SYKRAF1BRAFPDE4DPDE4A
SCHEMBL14320848 0.79 PDE4D (0.55) SYKRAF1BRAFPDE4DPDE4A
SCHEMBL30507985 0.79 KAT2B (0.50) SYKPDE4DPDE4APDE4BPDE4C
SCHEMBL25314851 0.79 KAT2B (0.50) SYKPDE4DPDE4APDE4BPDE4C
SCHEMBL18301635 0.79 SYK (0.41) SYKRAF1BRAFPDE4DPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019141131-A1 BROMODOMAIN INHIBITOR COMPOUND AND USE THEREOF 中国科学院上海药物研究所 2019-07-25 WO disclosed