SCHEMBL21200860

SCHEMBL21200860

COc1ccc2sc3ccccc3c(=O)c2c1Cl

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.72
RAB9A P51151 5/20 0.72
MAPT P10636 5/20 0.72
HPGD P15428 3/20 0.72
CYP1A2 P05177 1/20 0.72
CYP3A4 P08684 1/20 0.72
CYP2C9 P11712 1/20 0.72
CYP2C19 P33261 1/20 0.72
KDM4E B2RXH2 3/20 0.52
TDP1 Q9NUW8 3/20 0.52
ALDH1A1 P00352 3/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
KMT2A Q03164 4/20 0.46
MEN1 O00255 3/20 0.46
MAOA P21397 4/20 0.46
MAOB P27338 3/20 0.46
GAA P10253 2/20 0.43
POLB P06746 1/20 0.43
LMNA P02545 1/20 0.40
HCRTR1 O43613 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29936220 1.00 NPC1 (0.72) NPC1RAB9AMAPTHPGDCYP1A2
SCHEMBL29936580 0.85 MAPT (0.56) NPC1RAB9AMAPTHPGDCYP1A2
SCHEMBL21201163 0.85 MAPT (0.56) NPC1RAB9AMAPTHPGDCYP1A2
SCHEMBL942205 0.85 MAPT (0.56) NPC1RAB9AMAPTHPGDCYP1A2
SCHEMBL31157858 0.84 NPC1 (1.00) NPC1RAB9AMAPTHPGDCYP1A2
SCHEMBL22161850 0.84 NPC1 (0.74) NPC1RAB9AMAPTHPGDCYP1A2
SCHEMBL4306920 0.84 NPC1 (1.00) NPC1RAB9AMAPTHPGDCYP1A2
SCHEMBL29573388 0.82 MAPT (0.53) NPC1RAB9AMAPTHPGDCYP1A2
SCHEMBL148030 0.82 MAPT (0.53) NPC1RAB9AMAPTHPGDCYP1A2
SCHEMBL2789108 0.81 NPC1 (0.70) NPC1RAB9AMAPTHPGDCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 125 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250177927-A1 SUPPORTED MEMBRANES BY THERMAL AND UV INITITATED MASS POLYMERIZATION PROMERUS, LLC (US) 2025-06-05 US claimed
US-20250122402-A1 LONG SHELF-LIFE STABLE MASS POLYMERIZABLE POLYCYCLOOLEFIN COMPOSITIONS CONTAINING PYRIDINE LIGATED PALLADIUM COMPOUNDS PROMERUS, LLC (US) 2025-04-17 US claimed
EP-4437027-A1 DUAL UV BLOCKERS CONTAINING STABLE PHOTOACTIVE MASS POLYMERIZABLE POLYCYCLOOLEFIN COMPOSITIONS AS OPTICAL MATERIALS Promerus, LLC (US) 2024-10-02 EP claimed
US-20240254284-A1 UNSATURATED CYCLIC ANHYDRIDE END CAPPED POLYIMIDES AND POLYAMIC ACIDS AND PHOTOSENSITIVE COMPOSITIONS THEREOF PROMERUS, LLC (US) 2024-08-01 US claimed
WO-2024083874-A1 COMPOSITION MERCK PATENT GMBH (DE) 2024-04-25 WO claimed
EP-4087889-B1 STABLE MASS POLYMERIZABLE POLYCYCLOOLEFIN COMPOSITIONS AS 3D PRINTING MATERIALS AND A METHOD OF FABRICATION THEREOF PROMERUS LLC (US) 2024-03-06 EP claimed
US-11897991-B2 UV active derivatives of Pd(AcAc)2 catalyzed polycycloolefin compositions as optical materials PROMERUS, LLC (US) 2024-02-13 US claimed
EP-4288479-A1 LONG SHELF LIFE STABLE PHOTOACTIVE MASS POLYMERIZABLE POLYCYCLOOLEFIN COMPOSITIONS AS OPTICAL MATERIALS Promerus, LLC (US) 2023-12-13 EP claimed
US-11746166-B2 UV active derivatives of pd(AcAc)2L catalyzed polycycloolefin compositions as optical materials PROMERUS, LLC (US) 2023-09-05 US claimed
WO-2023158768-A1 DUAL CATALYST SYSTEM FOR MASS ROMP AND CATIONIC POLYMERIZABLE COMPOSITIONS PROMERUS, LLC (US) 2023-08-24 WO claimed
CN-111656792-B Polycycloolefin monomers as optical materials and catalysts activated by compounds capable of generating photoacid 住友电木株式会社 2022-03-15 CN claimed
US-20220010157-A1 HIGH IMPACT STRENGTH 3D PRINTING MATERIALS DERIVED FROM POLYCYCLOOLEFIN MONOMERS AND CROSSLINKERS PROMERUS, LLC (US) 2022-01-13 US claimed
WO-2021262921-A1 HINDERED AMINE STABILIZED UV ACTIVE ORGANOPALLADIUM CATALYZED POLYCYCLOOLEFIN COMPOSITIONS AS OPTICAL MATERIALS PROMERUS, LLC (US) 2021-12-30 WO claimed
WO-2021142402-A1 STABLE MASS POLYMERIZABLE POLYCYCLOOLEFIN COMPOSITIONS AS 3D PRINTING MATERIALS AND A METHOD OF FABRICATION THEREOF PROMERUS, LLC (US) 2021-07-15 WO claimed
WO-2021138651-A1 IMPROVED SHELF LIFE MASS POLYMERIZABLE POLYCYCLOOLEFIN COMPOSITIONS AS OPTICAL MATERIALS PROMERUS, LLC (US) 2021-07-08 WO claimed
US-20210198392-A1 UV ACTIVE DERIVATIVES OF Pd(AcAc)2 CATALYZED POLYCYCLOOLEFIN COMPOSITIONS AS OPTICAL MATERIALS PROMERUS, LLC (US) 2021-07-01 US claimed
CN-112335252-A Polycycloolefinic monomers as 3D printing materials and catalysts activated by compounds capable of generating photoacid 普罗米鲁斯有限责任公司 2021-02-05 CN claimed
US-20200283580-A1 UNSATURATED CYCLIC ANHYDRIDE END CAPPED POLYIMIDES AND POLYAMIC ACIDS AND PHOTOSENSITIVE COMPOSITIONS THEREOF PROMERUS, LLC (US) 2020-09-10 US claimed
WO-2020132665-A1 HIGH IMPACT STRENGTH 3D PRINTING MATERIALS DERIVED FROM POLYCYCOOLEFIN MONOMERS AND CROSSLINKERS PROMERUS, LLC (US) 2020-06-25 WO claimed
WO-2019147878-A1 POLYCYCLOOLEFIN MONOMERS AND CATALYST ACTIVATED BY COMPOUND CAPABLE OF GENERATING PHOTOACID AS OPTICAL MATERIALS PROMERUS, LLC (US) 2019-08-01 WO claimed