SCHEMBL21207261

SCHEMBL21207261

CCCCc1ccc2c(c1)NC(=O)CO2

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.74
NR3C2 P08235 3/20 0.58
MMP12 P39900 1/20 0.57
DRD4 P21917 6/20 0.51
DRD2 P14416 5/20 0.51
DRD3 P35462 3/20 0.51
ALDH1A1 P00352 3/20 0.51
MAPT P10636 2/20 0.49
MEN1 O00255 1/20 0.49
PSMD14 O00487 1/20 0.49
LMNA P02545 1/20 0.49
GAA P10253 1/20 0.49
HPGD P15428 1/20 0.49
XBP1 P17861 1/20 0.49
HTT P42858 1/20 0.49
KMT2A Q03164 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
HTR1A P08908 1/20 0.48
HTR1D P28221 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12844300 0.91 PARP1 (0.78) PARP1NR3C2MMP12DRD4DRD2
SCHEMBL31033201 0.91 PARP1 (0.78) PARP1NR3C2MMP12DRD4DRD2
SCHEMBL11004751 0.90 PARP1 (0.70) PARP1NR3C2MMP12DRD4DRD2
SCHEMBL11006154 0.90 PARP1 (0.70) PARP1NR3C2MMP12DRD4DRD2
SCHEMBL21177010 0.89 PARP1 (0.79) PARP1NR3C2MMP12DRD4DRD2
SCHEMBL11002313 0.88 PARP1 (0.77) PARP1NR3C2MMP12DRD4DRD2
SCHEMBL4178404 0.86 PARP1 (0.65) PARP1NR3C2MMP12DRD4DRD2
SCHEMBL9244955 0.86 PARP1 (0.65) PARP1NR3C2MMP12DRD4DRD2
SCHEMBL532134 0.85 PARP1 (1.00) PARP1NR3C2MMP12DRD4DRD2
SCHEMBL4257167 0.84 PARP1 (0.70) PARP1NR3C2MMP12DRD4DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019145919-A1 HETEROCYCLIC COMPOUNDS USEFUL AS ANTIBACTERIAL AGENTS CADILA HEALTHCARE LIMITED (IN) 2019-08-01 WO disclosed