SCHEMBL21208129

SCHEMBL21208129

Cc1nc2ccccn2c1-c1ccnc(N2CCNCC2)c1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CSNK1E P49674 1/20 0.47
ALDH1A1 P00352 1/20 0.47
POLB P06746 1/20 0.47
GAA P10253 1/20 0.47
MAPT P10636 1/20 0.47
NCOA1 Q15788 1/20 0.47
NCOA3 Q9Y6Q9 1/20 0.47
NMT1 P30419 10/20 0.47
KARS1 Q15046 2/20 0.47
DYRK1A Q13627 1/20 0.46
CDK4 P11802 1/20 0.46
CDK2 P24941 1/20 0.46
IRAK4 Q9NWZ3 1/20 0.44
TLR9 Q9NR96 1/20 0.44
TLR8 Q9NR97 1/20 0.44
TLR7 Q9NYK1 1/20 0.44
PLD1 Q13393 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21208130 0.88 CDK2 (0.48) ALDH1A1POLBGAAMAPTNCOA1
SCHEMBL21217063 0.86 PRKDC (0.52) CSNK1EALDH1A1POLBGAAMAPT
SCHEMBL21209372 0.85 CSNK1E (0.49) CSNK1ENMT1KARS1DYRK1ATLR9
SCHEMBL24688736 0.82 CSNK1E (0.56) CSNK1ENMT1KARS1DYRK1ATLR9
SCHEMBL21217032 0.80 IRAK4 (0.57) CSNK1EALDH1A1POLBGAAMAPT
SCHEMBL21208144 0.78 CDK2 (0.59) ALDH1A1POLBGAAMAPTNCOA1
SCHEMBL7965088 0.75 CDK2 (0.54) ALDH1A1POLBGAAMAPTNCOA1
SCHEMBL21209364 0.74 DRD1 (0.41) CSNK1EGAAMAPTNMT1CDK2
SCHEMBL3442456 0.73 DYRK1A (0.64) NMT1KARS1DYRK1APLD1
SCHEMBL9968482 0.72 MEN1 (0.52) ALDH1A1GAANMT1KARS1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019148136-A1 GCN2 INHIBITORS AND USES THEREOF MERCK PATENT GMBH (DE) 2019-08-01 WO disclosed