SCHEMBL21234205

SCHEMBL21234205

C[C@@H](O)[C@@H](C(N)=O)N1CC2(CCCN2C(=O)OC(C)(C)C)C1

nearest known ligand 0.64

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 1/20 0.64
GRIN2C Q14957 1/20 0.64
JAK3 P52333 4/20 0.40
SPR P35270 3/20 0.35
RET P07949 5/20 0.34
CNR2 P34972 1/20 0.32
TSHR P16473 1/20 0.32
NAMPT P43490 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18705165 0.84 GRIN2B (0.46) GRIN2BGRIN2CJAK3SPRRET
SCHEMBL21234082 0.83 GRIN2B (0.48) GRIN2BGRIN2CJAK3SPRRET
SCHEMBL21234076 0.83 GRIN2B (0.48) GRIN2BGRIN2CJAK3SPRRET
SCHEMBL21233783 0.83 GRIN2B (0.46) GRIN2BGRIN2CJAK3
SCHEMBL21234069 0.82 GRIN2B (0.45) GRIN2BGRIN2CJAK3
SCHEMBL21234128 0.81 GRIN2B (0.46) GRIN2BGRIN2CJAK3SPRRET
SCHEMBL18705161 0.80 JAK3 (0.44) GRIN2BGRIN2CJAK3SPRRET
SCHEMBL18705173 0.80 GRIN2B (0.46) GRIN2BGRIN2CJAK3SPRRET
SCHEMBL18705167 0.79 GRIN2B (0.45) GRIN2BGRIN2CJAK3SPRRET
Zelquistinel SCHEMBL24636775 0.78 GRIN2B (1.00) GRIN2BGRIN2CJAK3TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019152696-A1 SPIRO-LACTAM NMDA RECEPTOR MODULATORS AND USES THEREOF APTINYX INC. (US) 2019-08-08 WO disclosed