SCHEMBL21236859

SCHEMBL21236859

N#Cc1cc(CCO)cc(-c2ccc(Oc3ccc(F)cc3)cc2)n1

nearest known ligand 0.64

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 14/20 0.64
KDM4E B2RXH2 4/20 0.46
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
ALDH1A1 P00352 2/20 0.46
HPGD P15428 2/20 0.46
SQOR Q9Y6N5 1/20 0.45
LOXL2 Q9Y4K0 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL805915 0.90 SCN9A (0.67) SCN9AKDM4EMEN1KMT2AALDH1A1
SCHEMBL15383836 0.85 SCN9A (0.60) SCN9AKDM4EMEN1KMT2AALDH1A1
SCHEMBL21236837 0.78 SCN9A (0.72) SCN9A
SCHEMBL787725 0.78 SCN9A (1.00) SCN9A
SCHEMBL21236906 0.78 SCN9A (0.65) SCN9A
SCHEMBL787549 0.78 SCN9A (1.00) SCN9A
SCHEMBL787548 0.78 SCN9A (1.00) SCN9A
SCHEMBL805982 0.78 SCN9A (0.64) SCN9AKDM4EMEN1KMT2AALDH1A1
SCHEMBL806028 0.77 SCN9A (0.68) SCN9AKDM4EMEN1KMT2AALDH1A1
SCHEMBL805985 0.74 SCN9A (0.60) SCN9AKDM4EMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2616441-B1 PYRIDINE COMPOUNDS AND THE USES THEREOF PURDUE PHARMA LP (US) 2019-08-07 EP disclosed