SCHEMBL2123703

SCHEMBL2123703

CC(C)Nc1ccc(-c2nc(-c3ccc4c(c3)CCN(C(=O)C(NC(=O)O)C(C)(C)C)CC4)no2)cc1C#N

nearest known ligand 0.52

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 20/20 0.52
S1PR3 Q99500 9/20 0.52
KCNH2 Q12809 3/20 0.48
S1PR5 Q9H228 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3430626 0.89 S1PR1 (0.50) S1PR1S1PR3KCNH2S1PR5
SCHEMBL2123708 0.87 S1PR1 (0.69) S1PR1S1PR3KCNH2S1PR5
SCHEMBL2128462 0.85 S1PR1 (0.54) S1PR1S1PR3KCNH2
SCHEMBL2123723 0.85 S1PR1 (0.58) S1PR1S1PR3KCNH2S1PR5
SCHEMBL3430908 0.85 S1PR1 (0.55) S1PR1S1PR3KCNH2
SCHEMBL2125250 0.84 S1PR1 (0.57) S1PR1S1PR3KCNH2S1PR5
SCHEMBL2122355 0.83 S1PR1 (0.55) S1PR1S1PR3KCNH2
SCHEMBL2121432 0.83 S1PR1 (0.56) S1PR1S1PR3KCNH2S1PR5
SCHEMBL2122681 0.83 S1PR1 (0.60) S1PR1S1PR3KCNH2S1PR5
SCHEMBL2122728 0.83 S1PR1 (0.47) S1PR1S1PR3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2443110-A1 S1P1 AGONISTS COMPRISING A BICYCLIC N-CONTAINING RING Glaxo Group Limited (GB) 2012-04-25 EP disclosed
WO-2010146105-A1 S1P1 AGONISTS COMPRISING A BICYCLIC N-CONTAINING RING GLAXO GROUP LIMITED (GB) 2010-12-23 WO disclosed