SCHEMBL2124209

SCHEMBL2124209

Cc1c(-c2noc(-c3ccc(OC(C)C)c(C#N)c3)n2)ccc2c1CCN(C(=O)CCNC(=O)OCC(C)(C)C)C2

nearest known ligand 0.64

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 20/20 0.64
S1PR5 Q9H228 4/20 0.64
KCNH2 Q12809 3/20 0.62
CYP3A4 P08684 1/20 0.62
CYP2C9 P11712 1/20 0.62
S1PR3 Q99500 7/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13012484 0.92 S1PR1 (0.66) S1PR1S1PR5KCNH2CYP3A4CYP2C9
SCHEMBL3430872 0.91 S1PR1 (0.73) S1PR1S1PR5KCNH2CYP3A4CYP2C9
SCHEMBL2602069 0.89 S1PR1 (0.65) S1PR1S1PR5KCNH2CYP3A4CYP2C9
SCHEMBL2605724 0.89 S1PR1 (0.72) S1PR1S1PR5KCNH2CYP3A4CYP2C9
Hydrochloric Acid SCHEMBL2129274 0.88 S1PR1 (0.71) S1PR1S1PR5KCNH2CYP3A4CYP2C9
SCHEMBL3426267 0.88 S1PR1 (0.72) S1PR1S1PR5KCNH2CYP3A4CYP2C9
SCHEMBL2123002 0.86 S1PR1 (0.73) S1PR1S1PR5KCNH2CYP3A4CYP2C9
SCHEMBL2602070 0.86 S1PR1 (0.66) S1PR1S1PR5KCNH2CYP3A4CYP2C9
Hydrochloric Acid SCHEMBL2120921 0.85 S1PR1 (0.72) S1PR1S1PR5KCNH2CYP3A4CYP2C9
SCHEMBL3432043 0.85 S1PR1 (0.72) S1PR1S1PR5KCNH2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2443110-A1 S1P1 AGONISTS COMPRISING A BICYCLIC N-CONTAINING RING Glaxo Group Limited (GB) 2012-04-25 EP disclosed