SCHEMBL21242583

SCHEMBL21242583

O=C(Nc1nc2cccc(C3CCCCC3)n2n1)C1CC1

nearest known ligand 0.66

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
JAK1 P23458 19/20 0.66
JAK2 O60674 17/20 0.66
TYK2 P29597 16/20 0.66
JAK3 P52333 10/20 0.66
CYP2C19 P33261 2/20 0.66
CYP1A2 P05177 1/20 0.66
CYP2C9 P11712 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21242963 0.88 JAK1 (0.67) JAK1JAK2TYK2JAK3CYP2C19
SCHEMBL23766369 0.85 JAK1 (0.60) JAK1JAK2TYK2JAK3CYP2C19
SCHEMBL21242956 0.84 JAK1 (0.59) JAK1JAK2TYK2JAK3CYP2C19
SCHEMBL21757169 0.83 JAK2 (0.71) JAK1JAK2TYK2JAK3CYP2C19
SCHEMBL21757103 0.82 JAK2 (0.70) JAK1JAK2TYK2JAK3CYP2C19
SCHEMBL23424235 0.81 JAK2 (0.68) JAK1JAK2TYK2JAK3CYP2C19
SCHEMBL7966910 0.81 JAK1 (0.70) JAK1JAK2TYK2JAK3
SCHEMBL23080443 0.80 JAK1 (1.00) JAK1JAK2TYK2JAK3CYP2C19
SCHEMBL23766368 0.80 JAK2 (0.71) JAK1JAK2TYK2JAK3CYP2C19
SCHEMBL21242552 0.80 JAK1 (1.00) JAK1JAK2TYK2JAK3CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019149244-A1 JAK INHIBITOR AND USE THEREOF 南京明德新药研发股份有限公司 2019-08-08 WO disclosed