SCHEMBL21243058

SCHEMBL21243058

CC(C)c1cc(-c2ccncc2)c(-c2cccc3ccccc23)nn1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 10/20 0.65
MAPK11 Q15759 9/20 0.65
KDR P35968 4/20 0.45
CSNK1D P48730 7/20 0.44
KDM4E B2RXH2 1/20 0.43
NPC1 O15118 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
MAPK1 P28482 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HSD17B10 Q99714 1/20 0.43
MAPK13 O15264 1/20 0.39
GCGR P47871 1/20 0.39
MAPK12 P53778 1/20 0.39
TNF P01375 1/20 0.39
ALOX5 P09917 1/20 0.38
RIPK3 Q9Y572 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16092103 0.82 MAPK14 (0.70) MAPK14MAPK11KDRCSNK1DKDM4E
SCHEMBL17728180 0.81 MAPK14 (0.61) MAPK14MAPK11KDRCSNK1DKDM4E
SCHEMBL16092101 0.80 MAPK14 (0.66) MAPK14MAPK11KDRCSNK1DKDM4E
SCHEMBL16062323 0.80 MAPK14 (0.66) MAPK14MAPK11KDRCSNK1DKDM4E
SCHEMBL16092113 0.79 MAPK14 (1.00) MAPK14MAPK11KDRCSNK1DKDM4E
SCHEMBL16060785 0.79 MAPK14 (0.65) MAPK14MAPK11KDRCSNK1DKDM4E
SCHEMBL30360182 0.76 MAPK14 (0.76) MAPK14MAPK11KDRCSNK1DKDM4E
SCHEMBL21219601 0.76 MAPK14 (0.76) MAPK14MAPK11KDRCSNK1DKDM4E
SCHEMBL16092092 0.75 MAPK14 (0.60) MAPK14MAPK11KDRCSNK1DKDM4E
SCHEMBL30756642 0.74 TNF (0.63) MAPK14MAPK11KDM4ENPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3521284-A1 PYRAZINE COMPOUNDS AS MAP KINASE MODULATORS AND USES THEREOF The Trustees of Columbia University in the City of New York (US) 2019-08-07 EP disclosed