SCHEMBL2124806

SCHEMBL2124806

CCCNc1ncc(-c2nc(-c3ccc4c(c3)CCN(C(=O)CNC(=O)OC(C)(C)C)CC4)no2)cc1C#N

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 18/20 0.44
S1PR3 Q99500 6/20 0.44
KCNH2 Q12809 3/20 0.42
FNTA P49354 1/20 0.37
FNTB P49356 1/20 0.37
RET P07949 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2124233 0.90 S1PR1 (0.47) S1PR1S1PR3KCNH2RET
SCHEMBL2602093 0.90 S1PR1 (0.48) S1PR1S1PR3KCNH2
SCHEMBL2605713 0.90 FNTA (0.38) S1PR1S1PR3FNTAFNTB
SCHEMBL2605760 0.90 S1PR1 (0.47) S1PR1S1PR3KCNH2
SCHEMBL2602092 0.88 S1PR1 (0.48) S1PR1S1PR3KCNH2FNTAFNTB
SCHEMBL2602094 0.88 S1PR1 (0.49) S1PR1S1PR3KCNH2FNTAFNTB
SCHEMBL2124243 0.86 S1PR1 (0.47) S1PR1S1PR3KCNH2
Hydrochloric Acid SCHEMBL2123966 0.86 S1PR1 (0.47) S1PR1S1PR3KCNH2
SCHEMBL13012923 0.85 S1PR1 (0.52) S1PR1S1PR3KCNH2
SCHEMBL2123975 0.85 S1PR1 (0.54) S1PR1S1PR3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2443110-A1 S1P1 AGONISTS COMPRISING A BICYCLIC N-CONTAINING RING Glaxo Group Limited (GB) 2012-04-25 EP disclosed
WO-2010146105-A1 S1P1 AGONISTS COMPRISING A BICYCLIC N-CONTAINING RING GLAXO GROUP LIMITED (GB) 2010-12-23 WO disclosed