SCHEMBL21249985

SCHEMBL21249985

C=NC1=C(/C=C(\C)c2cc(NC(=O)c3ccnc(C(C)(F)F)c3)ccc2C)N2CCOC[C@H]2CC(=O)N1CC(C)(C)O

nearest known ligand 0.48

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 20/20 0.48
BRAF P15056 19/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21250042 0.79 RAF1 (0.47) RAF1BRAF
SCHEMBL19016613 0.78 RAF1 (0.61) RAF1BRAF
SCHEMBL21249948 0.78 RAF1 (0.48) RAF1BRAF
SCHEMBL19016103 0.75 RAF1 (0.60) RAF1BRAF
SCHEMBL23654041 0.75 RAF1 (0.53) RAF1BRAF
SCHEMBL21250036 0.74 RAF1 (0.46) RAF1BRAF
SCHEMBL19016388 0.74 RAF1 (0.52) RAF1BRAF
SCHEMBL19016015 0.73 RAF1 (0.65) RAF1BRAF
SCHEMBL19015977 0.73 RAF1 (0.65) RAF1BRAF
SCHEMBL19016060 0.73 RAF1 (0.65) RAF1BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10377770-B2 Tricyclic compounds and compositions as kinase inhibitors NOVARTIS AG (CH) 2019-08-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10377770-B2 Tricyclic compounds and compositions as kinase inhibitors BRAF, RAF1, MAP3K1 RAF1 2/4885BRAF 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.