SCHEMBL2125146

SCHEMBL2125146

Cc1c(-c2noc(-c3cnc(OC(C)C)c(C#N)c3)n2)ccc2c1CCN(C(=O)C(NC(=O)O)C(C)(C)C)C2

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 20/20 0.54
S1PR5 Q9H228 7/20 0.54
S1PR3 Q99500 8/20 0.53
KCNH2 Q12809 3/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2C9 P11712 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2125254 0.91 S1PR1 (0.49) S1PR1S1PR5S1PR3KCNH2CYP3A4
SCHEMBL13012566 0.88 S1PR1 (0.56) S1PR1S1PR5S1PR3KCNH2CYP3A4
SCHEMBL2130323 0.88 S1PR1 (0.55) S1PR1S1PR5S1PR3KCNH2CYP3A4
SCHEMBL2130329 0.88 S1PR1 (0.55) S1PR1S1PR5S1PR3KCNH2CYP3A4
SCHEMBL2123971 0.88 S1PR1 (0.55) S1PR1S1PR5S1PR3KCNH2CYP3A4
SCHEMBL2602085 0.87 S1PR1 (0.50) S1PR1S1PR5S1PR3KCNH2CYP3A4
Hydrochloric Acid SCHEMBL2122231 0.87 S1PR1 (0.54) S1PR1S1PR5S1PR3KCNH2CYP3A4
Hydrochloric Acid SCHEMBL2122226 0.87 S1PR1 (0.54) S1PR1S1PR5S1PR3KCNH2CYP3A4
SCHEMBL2130255 0.87 S1PR1 (0.52) S1PR1S1PR5S1PR3KCNH2CYP3A4
SCHEMBL2124514 0.87 S1PR1 (0.52) S1PR1S1PR5S1PR3KCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2443110-A1 S1P1 AGONISTS COMPRISING A BICYCLIC N-CONTAINING RING Glaxo Group Limited (GB) 2012-04-25 EP disclosed
WO-2010146105-A1 S1P1 AGONISTS COMPRISING A BICYCLIC N-CONTAINING RING GLAXO GROUP LIMITED (GB) 2010-12-23 WO disclosed