SCHEMBL21253013

SCHEMBL21253013

CC1(C)Cc2cc(C3=C(c4ccc(O[C@H]5CCN(CCCF)C5)cc4)c4ccc(C(=O)OF)cc4CCC3)ccc2N1

nearest known ligand 0.88

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 19/20 0.88
AGTR2 P50052 1/20 0.62
ESR2 Q92731 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19132049 0.95 ESR1 (0.88) ESR1AGTR2ESR2
SCHEMBL31739218 0.95 ESR1 (0.88) ESR1AGTR2ESR2
SCHEMBL24022268 0.95 ESR1 (0.88) ESR1AGTR2ESR2
SCHEMBL19154740 0.93 ESR1 (1.00) ESR1AGTR2ESR2
Hydrochloric Acid SCHEMBL19132002 0.93 ESR1 (0.99) ESR1AGTR2ESR2
SCHEMBL23336117 0.93 ESR1 (0.89) ESR1AGTR2ESR2
Hydrochloric Acid SCHEMBL29499972 0.93 ESR1 (0.99) ESR1AGTR2ESR2
SCHEMBL24022088 0.90 ESR1 (0.81) ESR1
SCHEMBL21253465 0.90 ESR1 (0.81) ESR1
SCHEMBL29499999 0.89 ESR1 (0.82) ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3524600-A1 PROCESSES AND INTERMEDIATES FOR THE PREPARATION OF NOVEL SUBSTITUTED 6,7-DIHYDRO-5H-BENZO[7]ANNULENE COMPOUNDS Sanofi (FR) 2019-08-14 EP disclosed