SCHEMBL2125342

SCHEMBL2125342

Cc1c(-c2noc(-c3cnc(OC(C)C)c(Cl)c3)n2)ccc2c1CCN(C(=O)O)C2C(C)(C)C

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 19/20 0.52
S1PR3 Q99500 9/20 0.52
S1PR5 Q9H228 4/20 0.52
MAP4K4 O95819 1/20 0.39
MINK1 Q8N4C8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2125913 0.91 S1PR1 (0.49) S1PR1S1PR3S1PR5
SCHEMBL2124893 0.89 S1PR1 (0.57) S1PR1S1PR3S1PR5MAP4K4MINK1
SCHEMBL2125344 0.87 S1PR1 (0.53) S1PR1S1PR3S1PR5MAP4K4MINK1
SCHEMBL3659387 0.82 S1PR1 (0.54) S1PR1S1PR3S1PR5
SCHEMBL13678374 0.82 S1PR1 (0.59) S1PR1S1PR3S1PR5
SCHEMBL2123481 0.81 S1PR1 (0.62) S1PR1S1PR3S1PR5
SCHEMBL3716238 0.80 S1PR1 (0.64) S1PR1S1PR3
SCHEMBL27669770 0.80 S1PR1 (0.56) S1PR1S1PR3S1PR5
SCHEMBL2122705 0.79 S1PR1 (0.50) S1PR1S1PR3S1PR5
SCHEMBL3753001 0.79 S1PR1 (0.46) S1PR1S1PR3S1PR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2443110-A1 S1P1 AGONISTS COMPRISING A BICYCLIC N-CONTAINING RING Glaxo Group Limited (GB) 2012-04-25 EP disclosed
WO-2010146105-A1 S1P1 AGONISTS COMPRISING A BICYCLIC N-CONTAINING RING GLAXO GROUP LIMITED (GB) 2010-12-23 WO disclosed