SCHEMBL2128247

SCHEMBL2128247

NC[C@H]1[C@@H]2CC[C@@H](C2)N1C(=O)c1nc(N2CCCC2)sc1-c1ccc(F)cc1

nearest known ligand 0.41

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 19/20 0.41
HCRTR2 O43614 16/20 0.41
HTR2A P28223 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2128241 0.86 NPC1 (0.40) HCRTR1HCRTR2HTR2A
SCHEMBL2128117 0.86 HCRTR1 (0.43) HCRTR1HCRTR2HTR2A
SCHEMBL2126486 0.83 HCRTR1 (0.44) HCRTR1HCRTR2
SCHEMBL2127485 0.83 HCRTR1 (0.44) HCRTR1HCRTR2
SCHEMBL2125951 0.81 HCRTR1 (0.43) HCRTR1HCRTR2
SCHEMBL2126406 0.80 HCRTR1 (0.42) HCRTR1HCRTR2
SCHEMBL982502 0.78 HCRTR1 (0.46) HCRTR1HCRTR2
SCHEMBL2126228 0.77 HCRTR1 (0.49) HCRTR1HCRTR2
SCHEMBL984110 0.75 HCRTR1 (0.41) HCRTR1HCRTR2
SCHEMBL2128177 0.75 HCRTR1 (0.56) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8236801-B2 2-aza-bicyclo[2.2.1]heptane derivatives ACTELION PHARMACEUTICALS LTD. (CH) 2012-08-07 US claimed
EP-2247586-B1 2-AZA-BICYCLO[2.2.1]HEPTANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2012-04-25 EP claimed
US-8236801-B2 2-aza-bicyclo[2.2.1]heptane derivatives ACTELION PHARMACEUTICALS LTD. (CH) 2012-08-07 US disclosed