SCHEMBL21285998

SCHEMBL21285998

Cn1cc(-c2ccc(NC(=O)C(NCCc3ccc(C#N)cc3)c3cccc(C(F)(F)F)c3)nc2)cn1

nearest known ligand 0.85

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
EP300 Q09472 20/20 0.85
CREBBP Q92793 1/20 0.79

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21285727 1.00 EP300 (0.85) EP300CREBBP
SCHEMBL23242143 1.00 EP300 (0.85) EP300CREBBP
SCHEMBL30011581 1.00 EP300 (0.85) EP300CREBBP
SCHEMBL21285895 0.92 EP300 (1.00) EP300CREBBP
SCHEMBL21286335 0.92 EP300 (1.00) EP300CREBBP
SCHEMBL23242099 0.92 EP300 (1.00) EP300CREBBP
SCHEMBL30011000 0.92 EP300 (1.00) EP300CREBBP
SCHEMBL23242128 0.91 EP300 (0.88) EP300CREBBP
SCHEMBL21285725 0.91 EP300 (0.88) EP300CREBBP
SCHEMBL21285729 0.91 EP300 (0.88) EP300CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3752497-B1 P300/CBP HAT INHIBITORS CONSTELLATION PHARMACEUTICALS INC (US) 2024-07-17 EP disclosed
US-20210115008-A1 P300/CBP HAT INHIBITORS CONSTELLATION PHARMACEUTICALS, INC. 2021-04-22 US disclosed
US-20210115008-A1 P300/CBP HAT INHIBITORS CONSTELLATION PHARMACEUTICALS, INC. 2021-04-22 US disclosed
WO-2021021893-A1 COMPOUNDS FOR USE IN TREATING NEUROLOGICAL DISORDERS CONSTELLATION PHARMACEUTICALS, INC. (US) 2021-02-04 WO disclosed
WO-2019161162-A1 P300/CBP HAT INHIBITORS CONSTELLATION PHARMACEUTICALS, INC. (US) 2019-08-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210115008-A1 P300/CBP HAT INHIBITORS EP300, HDAC1, KAT2A EP300 1/4885CREBBP 4/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.