SCHEMBL2128644

SCHEMBL2128644

COc1c(/C=C/c2ccc(NS(C)(=O)=O)cc2C(=O)O)cc(-c2ccc(C)[nH]c2=O)cc1C(C)(C)C

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.57
CRBN Q96SW2 1/20 0.39
FABP4 P15090 10/20 0.34
FABP5 Q01469 10/20 0.34
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
KMT2A Q03164 1/20 0.33
BRD4 O60885 1/20 0.32
PTPN5 P54829 1/20 0.32
FABP3 P05413 1/20 0.32
ATM Q13315 1/20 0.32
CHEK1 O14757 1/20 0.32
AURKA O14965 1/20 0.32
DAPK3 O43293 1/20 0.32
JAK2 O60674 1/20 0.32
ABL1 P00519 1/20 0.32
NTRK1 P04629 1/20 0.32
FYN P06241 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2128650 1.00 CYP3A4 (0.57) CYP3A4CRBNFABP4FABP5KDM4E
SCHEMBL2130343 0.93 CYP3A4 (0.57) CYP3A4CRBNHPGDBRD4CHEK1
SCHEMBL1543477 0.93 CYP3A4 (0.57) CYP3A4CRBNHPGDBRD4CHEK1
SCHEMBL2127429 0.92 CYP3A4 (0.57) CYP3A4CRBNFABP4FABP5PTPN5
SCHEMBL1542277 0.92 CYP3A4 (0.57) CYP3A4CRBNFABP4FABP5PTPN5
SCHEMBL2127426 0.87 CYP3A4 (0.76) CYP3A4CRBNFABP4FABP5PTPN5
SCHEMBL1542807 0.87 CYP3A4 (0.76) CYP3A4CRBNFABP4FABP5PTPN5
SCHEMBL2127697 0.86 CYP3A4 (0.75) CYP3A4CRBNBRD4
SCHEMBL2127702 0.86 CYP3A4 (0.75) CYP3A4CRBNBRD4
SCHEMBL2487208 0.86 CYP3A4 (0.56) CYP3A4CRBNFABP4FABP5PTPN5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2307372-B1 HETEROCYCLIC ANTIVIRAL COMPOUNDS HOFFMANN LA ROCHE (CH) 2012-04-25 EP claimed