SCHEMBL21338074

SCHEMBL21338074

C=CC(=C)Nc1cccc(Nc2nc(Nc3ccc(N[C@@H]4CCN(CCF)C4)cc3)ncc2F)c1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EGFR P00533 13/20 0.52
ITK Q08881 7/20 0.51
CCNT1 O60563 1/20 0.51
CCNE1 P24864 1/20 0.51
CDK2 P24941 1/20 0.51
CDK9 P50750 1/20 0.51
BTK Q06187 8/20 0.51
JAK3 P52333 1/20 0.51
ERBB2 P04626 1/20 0.49
ERBB3 P21860 1/20 0.49
ERBB4 Q15303 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16697962 0.92 EGFR (0.63) EGFRITKBTKJAK3ERBB2
SCHEMBL16391064 0.92 EGFR (0.63) EGFRITKBTKJAK3ERBB2
SCHEMBL16391059 0.92 EGFR (0.63) EGFRITKBTKJAK3ERBB2
SCHEMBL16391058 0.82 EGFR (0.67) EGFRITKBTKJAK3ERBB2
SCHEMBL16698236 0.82 EGFR (0.67) EGFRITKBTKJAK3ERBB2
SCHEMBL16391063 0.82 EGFR (0.67) EGFRITKBTKJAK3ERBB2
SCHEMBL16391055 0.80 EGFR (0.65) EGFRITKBTKJAK3ERBB2
SCHEMBL16371328 0.80 EGFR (0.65) EGFRITKBTKJAK3ERBB2
SCHEMBL16371329 0.80 EGFR (0.65) EGFRITKBTKJAK3ERBB2
SCHEMBL16391083 0.77 EGFR (0.78) EGFRITKBTKJAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3019496-B1 PYRIMIDINE DERIVATIVES AS KINASE INHIBITORS ACEA THERAPEUTICS INC (US) 2019-09-11 EP disclosed