SCHEMBL21345286

SCHEMBL21345286

Cc1ccc2c(c1)Oc1ccc(OC(F)(F)F)cc1NC2=O

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 19/20 0.61
TP53 P04637 1/20 0.52
POLB P06746 1/20 0.52
MAPT P10636 1/20 0.52
TDP1 Q9NUW8 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21345355 0.85 ABL1 (0.61) ABL1
SCHEMBL30437624 0.84 ABL1 (0.69) ABL1
SCHEMBL21345379 0.82 ABL1 (0.75) ABL1
SCHEMBL21333467 0.79 ABL1 (0.69) ABL1
SCHEMBL23296092 0.77 CES1 (0.77) ABL1
SCHEMBL31621242 0.77 CES1 (0.77) ABL1
SCHEMBL23191196 0.77 ABL1 (0.66) ABL1
SCHEMBL21333753 0.77 ABL1 (0.66) ABL1
SCHEMBL23191241 0.76 ABL1 (0.69) ABL1
SCHEMBL21346030 0.76 ABL1 (1.00) ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019173761-A1 C-ABL TYROSINE KINASE INHIBITORY COMPOUND EMBODIMENTS AND METHODS OF MAKING AND USING THE SAME THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2019-09-12 WO disclosed