SCHEMBL21363788

SCHEMBL21363788

CCCc1cc2c(cc1OCc1ccccc1)OCO2

nearest known ligand 0.55

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAOB P27338 4/20 0.55
MAOA P21397 3/20 0.46
TDP1 Q9NUW8 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
KMT2A Q03164 1/20 0.45
ALDH1A1 P00352 1/20 0.45
CYP3A4 P08684 1/20 0.45
TSHR P16473 1/20 0.45
GAA P10253 1/20 0.43
HTR1A P08908 1/20 0.43
DRD2 P14416 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
PDE5A O76074 1/20 0.42
EDNRB P24530 1/20 0.42
EDNRA P25101 1/20 0.42
MAPT P10636 1/20 0.41
MAPK1 P28482 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21363672 0.92 MAOB (0.52) MAOBMAOATDP1L3MBTL1KMT2A
SCHEMBL21363757 0.89 MAOB (0.50) MAOBMAOATDP1L3MBTL1KMT2A
SCHEMBL21366597 0.88 MAOB (0.57) MAOBMAOATDP1L3MBTL1KMT2A
SCHEMBL14552343 0.83 MAOB (0.52) MAOBMAOATDP1L3MBTL1KMT2A
SCHEMBL9292582 0.82 MAOB (0.51) MAOBMAOATDP1L3MBTL1KMT2A
Hydrochloric Acid SCHEMBL9293053 0.81 MAOB (0.50) MAOBMAOATDP1L3MBTL1KMT2A
SCHEMBL13854257 0.81 MAOB (0.59) MAOBMAOATDP1L3MBTL1KMT2A
SCHEMBL21363607 0.80 MAOB (0.51) MAOBMAOATDP1L3MBTL1KMT2A
SCHEMBL14552348 0.79 MAOB (0.54) MAOBMAOATDP1L3MBTL1KMT2A
SCHEMBL9789581 0.78 MAOB (0.59) MAOBMAOATDP1L3MBTL1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019175712-A1 NEW USES FOR CATECHOL MOLECULES AS INHIBITORS TO GLUTATHIONE S-TRANSFERASE METABOLIC PATHWAYS BASF CORPORATION (US) 2019-09-19 WO disclosed
WO-2019175713-A1 NEW CATECHOL MOLECULES AND THEIR USE AS INHIBITORS TO P450 RELATED METABOLIC PATHWAYS BASF CORPORATION (US) 2019-09-19 WO disclosed