SCHEMBL21367370

SCHEMBL21367370

Cc1ccc(NC(=O)c2ccc(CN3CCN(C)CC3)c(C)c2)cc1C#Cc1cnc2cccnn12

nearest known ligand 0.85

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 18/20 0.85
ABL2 P42684 2/20 0.84
CYP3A4 P08684 6/20 0.82
KCNH2 Q12809 6/20 0.82
LCK P06239 2/20 0.82
SRC P12931 2/20 0.82
PDGFRA P16234 2/20 0.82
EPHB2 P29323 2/20 0.82
EPHB3 P54753 2/20 0.82
EPHB4 P54760 2/20 0.82
DDR2 Q16832 2/20 0.82
GAK O14976 1/20 0.82
MLNR O43193 1/20 0.82
RIPK2 O43353 1/20 0.82
JAK2 O60674 1/20 0.82
NR1I2 O75469 1/20 0.82
ABCB11 O95342 1/20 0.82
MAP4K4 O95819 1/20 0.82
EGFR P00533 1/20 0.82
NR3C1 P04150 1/20 0.82

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13194694 0.97 ABL1 (0.88) ABL1ABL2CYP3A4KCNH2LCK
SCHEMBL16644576 0.93 ABL1 (0.82) ABL1ABL2CYP3A4KCNH2LCK
SCHEMBL15242137 0.93 ABL1 (0.85) ABL1ABL2CYP3A4KCNH2LCK
SCHEMBL12989619 0.92 ABL1 (1.00) ABL1ABL2CYP3A4KCNH2LCK
SCHEMBL589689 0.92 ABL1 (1.00) ABL1ABL2CYP3A4KCNH2LCK
SCHEMBL591027 0.91 ABL1 (1.00) ABL1ABL2CYP3A4KCNH2LCK
SCHEMBL15473029 0.91 ABL1 (0.83) ABL1ABL2CYP3A4KCNH2LCK
SCHEMBL24123124 0.91 ABL1 (1.00) ABL1ABL2CYP3A4KCNH2LCK
SCHEMBL588806 0.90 ABL1 (1.00) ABL1ABL2CYP3A4KCNH2LCK
Ponatinib SCHEMBL589260 0.90 ABL1 (1.00) ABL1ABL2CYP3A4KCNH2LCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019161495-A9 RIPK2 INHIBITORS THE GOVERNORS OF THE UNIVERSITY OF ALBERTA (CA) 2019-09-19 WO disclosed