SCHEMBL21369917

SCHEMBL21369917

OC(CN1CCCCC1)c1ccc2c(c1)CCc1c-2noc1-c1noc(-c2ccccc2)c1C(F)(F)F

nearest known ligand 0.68

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 20/20 0.68
S1PR3 Q99500 17/20 0.68
CYP3A4 P08684 1/20 0.50
CYP2C8 P10632 1/20 0.50
KCNH2 Q12809 1/20 0.50
S1PR4 O95977 1/20 0.46
S1PR5 Q9H228 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12000504 0.88 S1PR1 (0.89) S1PR1S1PR3CYP3A4CYP2C8KCNH2
SCHEMBL12000505 0.88 S1PR1 (0.89) S1PR1S1PR3CYP3A4CYP2C8KCNH2
SCHEMBL1812433 0.88 S1PR1 (0.89) S1PR1S1PR3CYP3A4CYP2C8KCNH2
SCHEMBL1813133 0.87 S1PR1 (0.63) S1PR1S1PR3CYP3A4CYP2C8KCNH2
SCHEMBL12000514 0.86 S1PR1 (0.89) S1PR1S1PR3CYP2C8KCNH2S1PR4
SCHEMBL12000515 0.86 S1PR1 (0.89) S1PR1S1PR3CYP2C8KCNH2S1PR4
SCHEMBL1810489 0.86 S1PR1 (0.89) S1PR1S1PR3CYP2C8KCNH2S1PR4
SCHEMBL1813155 0.83 S1PR1 (0.64) S1PR1S1PR3CYP3A4CYP2C8KCNH2
SCHEMBL21369960 0.83 S1PR1 (0.75) S1PR1S1PR3CYP3A4CYP2C8KCNH2
SCHEMBL1815203 0.83 S1PR1 (0.65) S1PR1S1PR3CYP3A4CYP2C8KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2592071-B1 Tricyclic heterocyclic compounds BRISTOL MYERS SQUIBB CO (US) 2019-09-18 EP disclosed